SCHEMBL11375973

SCHEMBL11375973

CC1=C(C(=O)C(=O)O)c2ccccc2CN1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
CLK4 Q9HAZ1 2/20 0.34
DYRK1B Q9Y463 2/20 0.34
TYRO3 Q06418 1/20 0.34
NTRK2 Q16620 1/20 0.34
HSD17B3 P37058 1/20 0.34
PARP1 P09874 2/20 0.33
KDM4E B2RXH2 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
SRD5A2 P31213 2/20 0.32
SRD5A1 P18405 1/20 0.32
PDPK1 O15530 1/20 0.32
PARP10 Q53GL7 1/20 0.32
PARP11 Q9NR21 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
FYN P06241 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10956402 0.75 SRD5A2 (0.41) KDM4ESRD5A2SMN1; SMN2CES1ALDH1A1
SCHEMBL21508269 0.71 CA12 (0.52) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL11155843 0.70 KDM4E (0.37) KDM4EALOX15TSHRSIRT1L3MBTL1
Bicarbonate SCHEMBL29928922 0.68 CA12 (0.84) CA12CA9CLK4DYRK1BTYRO3
Bicarbonate SCHEMBL21081705 0.68 CA12 (0.84) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL3373516 0.68 CA12 (0.53) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL3371700 0.67 CA12 (0.56) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL28209349 0.65 CA12 (0.62) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL12629638 0.65 CA12 (0.48) CA12CA9CLK4DYRK1BTYRO3
SCHEMBL14424495 0.63 CA12 (0.47) CA12CA9CLK4DYRK1BTYRO3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0030861-A2 Isoquinoline acetic acids and pharmaceutical compositions thereof PFIZER INC. (US) 1981-06-24 EP disclosed