SCHEMBL11385992

SCHEMBL11385992

CCCc1ncccc1C#N.c1cc2ccc1-2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.46
ALDH1A1 P00352 5/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
NPC1 O15118 4/20 0.45
RAB9A P51151 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
CASP3 P42574 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
ELANE P08246 2/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7213726 0.95 HPGD (0.49) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL7219978 0.85 HPGD (0.56) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL3313973 0.83 HPGD (0.51) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL30805704 0.82 HPGD (0.50) HPGDALDH1A1L3MBTL1KDM4EGAA
Hydrochloric Acid SCHEMBL28530423 0.81 HPGD (0.49) HPGDALDH1A1L3MBTL1KDM4EGAA
Hydrochloric Acid SCHEMBL30805705 0.81 HPGD (0.49) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL3791629 0.80 HPGD (0.51) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL4062196 0.77 ALDH1A1 (0.41) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL27933237 0.77 HPGD (0.39) HPGDALDH1A1L3MBTL1KDM4EGAA
SCHEMBL11370703 0.75 KDM4E (0.56) HPGDALDH1A1L3MBTL1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4260759-A CONDENSATION OF NITRILES SCHERING-CORPORATION (US) 1981-04-07 US disclosed
US-4115395-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1978-09-19 US disclosed
US-4107166-A ANTIFUNGAL, ANTIBACTERIAL SCHERING CORPORATION (US) 1978-08-15 US disclosed
US-4017500-A FUNGICIDES, BACTERICIDES SCHERING CORPORATION (US) 1977-04-12 US disclosed