SCHEMBL11387752

SCHEMBL11387752

OCc1cc2c3ccccc3[nH]c(=S)n2n1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
ADORA3 P0DMS8 9/20 0.40
PDE7A Q13946 1/20 0.38
PDE7B Q9NP56 1/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.37
PRNP P04156 1/20 0.37
HPGD P15428 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pirquinozol SCHEMBL635679 0.83 ADORA3 (0.59) ALDH1A1ADORA3
SCHEMBL11406627 0.80 ADORA3 (0.47) ALDH1A1ADORA3
SCHEMBL11392211 0.76 ADORA3 (0.54) ALDH1A1ADORA3PDE7APDE7BKMT2A
SCHEMBL11254079 0.72 ADORA3 (0.56) ALDH1A1ADORA3HPGD
SCHEMBL11391453 0.72 ADORA3 (0.77) ALDH1A1ADORA3KMT2AKDM4EMEN1
SCHEMBL31461654 0.71 SMN1; SMN2 (0.43) ALDH1A1ADORA3KMT2AKDM4EMEN1
SCHEMBL11395024 0.69 PDE7A (0.44) ALDH1A1ADORA3PDE7APDE7BKMT2A
SCHEMBL16370935 0.69 PDE7A (0.44) ALDH1A1PDE7APDE7BKMT2AKDM4E
SCHEMBL11288740 0.69 ADORA3 (0.56) ADORA3
SCHEMBL11250103 0.69 ADORA3 (0.58) ALDH1A1ADORA3KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4282226-A Thioxopyrazolo[1,5-c]quinazoline derivatives, anti-allergic compositions and methods for treating allergic conditions by parenteral administration, aerosol or insufflation E. R. SQUIBB & SONS, INC. (US) 1981-08-04 US disclosed