SCHEMBL11398596

SCHEMBL11398596

O=c1ccc2cccc3c2n1CO3

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.36
DRD2 P14416 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
CA12 O43570 1/20 0.32
BRD4 O60885 1/20 0.32
BRPF1 P55201 1/20 0.32
CA9 Q16790 1/20 0.32
KAT2B Q92831 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
TYMS P04818 1/20 0.32
MCL1 Q07820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15828537 0.81 ALDH1A1 (0.39) HTR1ADRD2KDM4ECA12BRD4
SCHEMBL3785969 0.70 HTR1A (0.41) HTR1ADRD2KDM4EMAPT
SCHEMBL19751542 0.67 ALDH1A1 (0.32)
SCHEMBL4999235 0.67 HTR1A (0.38) HTR1ADRD2KDM4EMAPTCA12
SCHEMBL4421682 0.66 HTR1A (0.46) HTR1ADRD2KDM4EMAPTMCL1
SCHEMBL10967544 0.65 CA12 (0.41) HTR1ADRD2KDM4ECA12BRD4
SCHEMBL4357253 0.65 CA12 (0.38) HTR1ADRD2KDM4ECA12BRD4
Oxirane SCHEMBL865844 0.64 KDM4E (0.31) KDM4ETYMS
SCHEMBL5982877 0.64 HTR1A (0.36) HTR1ADRD2CA12BRD4BRPF1
SCHEMBL11207376 0.63 HPGD (0.55) HTR1ADRD2KDM4EMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4251534-A Antihypertensive polyfluorohydroxyisopropyl bicyclic and tricyclic carbostyrils E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-02-17 US disclosed