SCHEMBL113998

SCHEMBL113998

Cc1cc(C)n(C(C=O)N2CCN(c3ccc(F)cc3-c3cnc(N4CCOCC4)nc3)CC2)n1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 4/20 0.39
WDR5 P61964 11/20 0.38
PIK3CA P42336 1/20 0.37
MTOR P42345 1/20 0.37
CNR2 P34972 1/20 0.37
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
TNIK Q9UKE5 1/20 0.36
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113873 0.90 KDM4E (0.41) WDR5TNIK
SCHEMBL112035 0.90 CNR2 (0.42) AOC3WDR5CNR2ALOX5APFEN1
SCHEMBL114572 0.85 DHFR (0.33) PIK3CATNIKLRRK2
SCHEMBL113125 0.83 CXCR3 (0.40) AOC3CNR2ALOX5APFEN1
SCHEMBL114041 0.82 CXCR3 (0.39) AOC3FEN1
SCHEMBL113141 0.82 CXCR3 (0.38) AOC3WDR5CNR2ALOX5APFEN1
SCHEMBL114405 0.80 CXCR3 (0.39) AOC3
SCHEMBL113179 0.80 CNR2 (0.40) AOC3WDR5CNR2ALOX5APFEN1
SCHEMBL114021 0.79 CXCR3 (0.37) ALOX5APFEN1
SCHEMBL112171 0.79 CNR2 (0.48) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed