SCHEMBL11400630

SCHEMBL11400630

CC1C(=O)NC2=Nc3cccc(Br)c3CN21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 9/20 0.73
PDE3A Q14432 9/20 0.73
LMNA P02545 1/20 0.73
CYP1A2 P05177 1/20 0.73
CYP3A4 P08684 1/20 0.73
CYP2D6 P10635 1/20 0.73
TSHR P16473 1/20 0.73
BLM P54132 1/20 0.73
PIM1 P11309 1/20 0.31
CSNK1A1 P48729 1/20 0.31
CDK5 Q00535 1/20 0.31
ROCK1 Q13464 1/20 0.31
DYRK1A Q13627 1/20 0.31
LRRK2 Q5S007 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
MEN1 O00255 1/20 0.31
PDE2A O00408 1/20 0.31
KMT2A Q03164 1/20 0.31
P2RY12 Q9H244 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11158019 0.85 PDE3B (0.74) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL2463520 0.84 PDE3B (1.00) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL120976 0.84 PDE3B (1.00) PDE3BPDE3ALMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11280120 0.84 PDE3B (0.73) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL9718399 0.83 PDE3B (1.00) PDE3BPDE3ALMNACYP1A2CYP3A4
Quazinone SCHEMBL11279841 0.83 PDE3B (0.97) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL11391653 0.82 PDE3B (0.76) PDE3BPDE3ALMNACYP1A2CYP3A4
Bromide SCHEMBL11168072 0.82 PDE3B (0.97) PDE3BPDE3ALMNACYP1A2CYP3A4
SCHEMBL11273531 0.78 PDE3B (0.64) PDE3BPDE3ALMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL11281642 0.77 PDE3B (0.62) PDE3BPDE3ALMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4256748-A INOTROPIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1981-03-17 US disclosed