SCHEMBL11405384

SCHEMBL11405384

Cn1nc(N)nc1NCCC(CN1CCCCC1)Oc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.36
KAT2B Q92831 2/20 0.36
CYP2D6 P10635 2/20 0.36
TSHR P16473 1/20 0.36
HIF1A Q16665 1/20 0.36
MCHR1 Q99705 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HRH3 Q9Y5N1 6/20 0.34
SLC6A4 P31645 4/20 0.34
SLC6A2 P23975 2/20 0.34
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
TRPC5 Q9UL62 1/20 0.33
DRD4 P21917 1/20 0.33
CCKAR P32238 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD3 P35462 1/20 0.33
SCN1A P35498 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27589491 0.75 ACHE (0.42) LTA4HCYP2D6TSHRHIF1AMCHR1
SCHEMBL9643684 0.74 HRH2 (0.51) LTA4HCYP2D6TSHRHIF1AKDM4E
SCHEMBL28354366 0.73 CYP2D6 (0.50) LTA4HCYP2D6TSHRHIF1AKDM4E
Lamtidine SCHEMBL534965 0.70 HRH2 (0.61) CYP2D6TSHRHIF1AHRH3LMNA
SCHEMBL11098343 0.69 HRH2 (0.56) CYP2D6TSHRHIF1AHRH3LMNA
SCHEMBL8813882 0.66 LTA4H (0.54) LTA4HCYP2D6TSHRHIF1AKDM4E
SCHEMBL11121993 0.65 HRH2 (0.45) CYP2D6TSHRHIF1AHRH3LMNA
SCHEMBL10672622 0.64 KDM4E (0.30) KDM4E
SCHEMBL11093148 0.62 HRH3 (0.33) CYP2D6TSHRHIF1AHRH3CYP1A2
SCHEMBL6052629 0.61 HRH3 (0.48) TSHRKDM4EHRH3SLC6A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0057564-A1 Process for preparing 3,5-diamino-1,2,4-triazoles SMITHKLINE BECKMAN CORPORATION (US) 1982-08-11 EP disclosed