SCHEMBL11407482

SCHEMBL11407482

N#CC(O)C(N)Cc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.52
SLC6A2 P23975 2/20 0.48
SLC6A3 Q01959 2/20 0.48
CTSC P53634 1/20 0.47
DPP4 P27487 2/20 0.40
FAP Q12884 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
ACACB O00763 1/20 0.38
CYP2D6 P10635 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
HTR2B P41595 1/20 0.36
CHRNA4 P43681 1/20 0.36
ESR1 P03372 3/20 0.36
ESR2 Q92731 3/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11424125 0.84 ESR1 (0.53) SLC6A2CYP1A2CYP2C19ESR1ESR2
SCHEMBL11407228 0.84 ESR1 (0.53) SLC6A2CYP1A2CYP2C19ESR1ESR2
SCHEMBL11411311 0.82 DPP4 (0.40) SLC6A2CTSCDPP4FAPDPP8
SCHEMBL11412673 0.81 EPHX1 (0.48) SLC6A4SLC6A2SLC6A3CTSCTAAR1
SCHEMBL8690443 0.81 EPHX1 (0.48) SLC6A4SLC6A2SLC6A3CTSCTAAR1
SCHEMBL11405363 0.78 SLC6A4 (0.54) SLC6A4DPP4FAPDPP8DPP9
SCHEMBL18703964 0.77 SLC6A4 (0.48) SLC6A4SLC6A2SLC6A3CTSCDPP4
SCHEMBL10763436 0.74 SLC6A4 (0.67) SLC6A4SLC6A2SLC6A3CYP2D6CYP1A2
SCHEMBL6357746 0.73 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3CYP2D6CYP2C19
SCHEMBL5812524 0.73 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4240975-A USED AS ENZYME INHIBITOR, ANTIFERTILITY AGENT, AND ENHANCES THE ANTITUMOR EFFECT OF BLEOMYCIN ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1980-12-23 US disclosed
US-4189604-A PEPTIDASE ENZYME INHIBITORS ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1980-02-19 US disclosed