SCHEMBL8690443

SCHEMBL8690443

N#CC(O)C(N)Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.48
ANPEP P15144 5/20 0.48
CTSC P53634 4/20 0.47
SLC15A1 P46059 1/20 0.47
CSNK1E P49674 1/20 0.46
ALPI P09923 1/20 0.46
PKM P14618 1/20 0.46
PTGS1 P23219 1/20 0.46
XIAP P98170 1/20 0.46
SLC7A5 Q01650 1/20 0.46
SLC6A2 P23975 2/20 0.45
TAAR1 Q96RJ0 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
LAP3 P28838 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11412673 1.00 EPHX1 (0.48) EPHX1ANPEPCTSCSLC15A1CSNK1E
SCHEMBL11412914 0.85 LTA4H (0.62) PTGS1SLC6A2MAOASLC6A3LAP3
SCHEMBL11424125 0.83 ESR1 (0.53) SLC7A5SLC6A2TAAR1
SCHEMBL11407228 0.83 ESR1 (0.53) SLC7A5SLC6A2TAAR1
SCHEMBL11411311 0.81 DPP4 (0.40) ANPEPCTSCSLC6A2TAAR1CYP2A6
SCHEMBL11407482 0.81 SLC6A4 (0.52) CTSCSLC6A2TAAR1SLC6A4SLC6A3
SCHEMBL11025286 0.81 SLC15A1 (0.51) EPHX1ANPEPSLC15A1CSNK1EALPI
SCHEMBL6580781 0.81 SLC15A1 (0.51) EPHX1ANPEPSLC15A1CSNK1EALPI
SCHEMBL6243841 0.81 SLC15A1 (0.51) EPHX1ANPEPSLC15A1CSNK1EALPI
SCHEMBL10431094 0.78 CSNK1E (0.51) EPHX1ANPEPCTSCSLC15A1CSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188106-A Process for preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO (JP) 1998-07-22 CN claimed
EP-0849257-A1 Process for the preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO., LTD. (JP) 1998-06-24 EP claimed
US-5834618-A CHEMICAL INTERMEDIATE FOR PROTEASE INHIBITOR DRUG KURARAY CO., LTD. (JP) 1998-11-10 US disclosed
US-5834618-A CHEMICAL INTERMEDIATE FOR PROTEASE INHIBITOR DRUG KURARAY CO., LTD. (JP) 1998-11-10 US disclosed
US-5834618-A CHEMICAL INTERMEDIATE FOR PROTEASE INHIBITOR DRUG KURARAY CO., LTD. (JP) 1998-11-10 US disclosed
CN-1188106-A Process for preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO (JP) 1998-07-22 CN disclosed
CN-1188106-A Process for preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO (JP) 1998-07-22 CN disclosed
CN-1188106-A Process for preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO (JP) 1998-07-22 CN disclosed
EP-0849257-A1 Process for the preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO., LTD. (JP) 1998-06-24 EP disclosed
EP-0849257-A1 Process for the preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO., LTD. (JP) 1998-06-24 EP disclosed
EP-0849257-A1 Process for the preparation of 3-amino-2-hydroxy-4-phenylbutyronitrile derivatives KURARAY CO., LTD. (JP) 1998-06-24 EP disclosed
US-4240975-A USED AS ENZYME INHIBITOR, ANTIFERTILITY AGENT, AND ENHANCES THE ANTITUMOR EFFECT OF BLEOMYCIN ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1980-12-23 US disclosed
US-4189604-A PEPTIDASE ENZYME INHIBITORS ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1980-02-19 US disclosed