SCHEMBL11414780

SCHEMBL11414780

COC(=O)C(C)CC(CC(CC(CCC(=O)O)C(=O)OC)C(=O)OC)C(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.44
GABRP O00591 2/20 0.39
GABRD O14764 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB1 P18505 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA3 P34903 2/20 0.39
GABRA2 P47869 2/20 0.39
GABRB2 P47870 2/20 0.39
GABRA4 P48169 2/20 0.39
GABRE P78334 2/20 0.39
GABRA6 Q16445 2/20 0.39
GABRG1 Q8N1C3 2/20 0.39
GABRG3 Q99928 2/20 0.39
GABRQ Q9UN88 2/20 0.39
NAALAD2 Q9Y3Q0 1/20 0.39
FOLH1 Q04609 11/20 0.39
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3273833 0.85 MME (0.47) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL1419634 0.85 MME (0.47) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL3275556 0.85 MME (0.47) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL712283 0.81 CYP1A2 (0.60) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL10254859 0.81 CYP1A2 (0.60) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL11986003 0.77 CA1 (0.52) CA1CA2SLC1A1
SCHEMBL19428729 0.77 CA1 (0.52) CA1CA2SLC1A1
SCHEMBL28267007 0.77 CA1 (0.62) CYP1A2GABRPGABRDGABRA1GABRB1
SCHEMBL12914922 0.77 CA1 (0.52) CA1CA2SLC1A1
SCHEMBL9609800 0.77 CA1 (0.52) CA1CA2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4242228-A URANIUM COMPOUND, ALKALI METAL COMPOUND, HALIDE AND DIHALOBUTENE AND/OR CARBOXYLIC ACID PHILLIPS PETROLEUM COMPANY (US) 1980-12-30 US claimed
US-4237312-A ACYCLIC CONJUGATED DIOLEFIN ESTRIFIED BY A CARBOXYLIC ACID IN A COPPER OR ANTIMONY COMPOUND CATALYST PHILLIPS PETROLEUM COMPANY (US) 1980-12-02 US claimed
US-4221917-A IODOSOARYL DICARBOXYLATE CATALYST PHILLIPS PETROLEUM COMPANY (US) 1980-09-09 US claimed
US-4216119-A IN A CARBOXYLIC ACID MEDIA PHILLIPS PETROLEUM COMPANY (US) 1980-08-05 US claimed
US-4213879-A HYDROCARBYL TITANIUM COMPOUND OR HYDROCARBYL TITANIUM HALIDE PROVE USEFUL IN THE OXIDATION OF CONJUGATED DIOLEFINS TO DIACYLOXY OLEFINS PHILLIPS PETROLEUM COMPANY (US) 1980-07-22 US claimed
US-4180676-A Conversion of conjugated diolefins to diacyloxy olefins PHILLIPS PETROLEUM COMPANY (US) 1979-12-25 US claimed
US-4164615-A USING AS CATALYST A TITANIUM COMPOUND, AN ALKALI METAL COMPOUND, AND A HALIDE PHILLIPS PETROLEUM COMPANY (US) 1979-08-14 US claimed
US-4162363-A BY REACTION WITH OXYGEN AND A CARBOXYLIC ACID COMPONENT PHILLIPS PETROLEUM COMPANY (US) 1979-07-24 US claimed
US-4242228-A URANIUM COMPOUND, ALKALI METAL COMPOUND, HALIDE AND DIHALOBUTENE AND/OR CARBOXYLIC ACID PHILLIPS PETROLEUM COMPANY (US) 1980-12-30 US disclosed
US-4237312-A ACYCLIC CONJUGATED DIOLEFIN ESTRIFIED BY A CARBOXYLIC ACID IN A COPPER OR ANTIMONY COMPOUND CATALYST PHILLIPS PETROLEUM COMPANY (US) 1980-12-02 US disclosed
US-4216119-A IN A CARBOXYLIC ACID MEDIA PHILLIPS PETROLEUM COMPANY (US) 1980-08-05 US disclosed
US-4213879-A HYDROCARBYL TITANIUM COMPOUND OR HYDROCARBYL TITANIUM HALIDE PROVE USEFUL IN THE OXIDATION OF CONJUGATED DIOLEFINS TO DIACYLOXY OLEFINS PHILLIPS PETROLEUM COMPANY (US) 1980-07-22 US disclosed
US-4180676-A Conversion of conjugated diolefins to diacyloxy olefins PHILLIPS PETROLEUM COMPANY (US) 1979-12-25 US disclosed
US-4164615-A USING AS CATALYST A TITANIUM COMPOUND, AN ALKALI METAL COMPOUND, AND A HALIDE PHILLIPS PETROLEUM COMPANY (US) 1979-08-14 US disclosed
US-4162363-A BY REACTION WITH OXYGEN AND A CARBOXYLIC ACID COMPONENT PHILLIPS PETROLEUM COMPANY (US) 1979-07-24 US disclosed