SCHEMBL11418985

SCHEMBL11418985

COC(=O)c1ccc(C=Nc2c(Cl)cccc2Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
PTGS2 P35354 2/20 0.51
PTGS1 P23219 1/20 0.51
MAPT P10636 3/20 0.50
ALDH1A1 P00352 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRIN2B Q13224 1/20 0.50
GRIN2C Q14957 1/20 0.50
GRIN3A Q8TCU5 1/20 0.50
MAPK1 P28482 1/20 0.50
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11418984 1.00 CA1 (0.58) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11415368 0.87 CA1 (0.56) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11415365 0.87 CA1 (0.56) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11418549 0.85 CA1 (0.55) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11418552 0.85 CA1 (0.55) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11409392 0.84 CA1 (0.62) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11409395 0.84 CA1 (0.62) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11416460 0.83 CA1 (0.53) CA1CA2PTGS2PTGS1MAPT
SCHEMBL11416463 0.83 CA1 (0.53) CA1CA2PTGS2PTGS1MAPT
SCHEMBL13934092 0.78 CA2 (0.88) CA1CA2PTGS2PTGS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4200648-A INFLAMMATION BY ADMINISTERING A BENZYLIDENEANILINE DERIVATIVE WILLIAM H. RORER, INC. (US) 1980-04-29 US disclosed
US-4198349-A ANTIINFLAMMATORY, TOPICAL WILLIAM H. RORER, INC. (US) 1980-04-15 US disclosed