SCHEMBL11427741

SCHEMBL11427741

NC(=O)c1cc(C(O)CN2CCC(n3c(=O)[nH]c4ccccc43)CC2)ccc1O

nearest known ligand 0.98

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 10/20 0.98
ADRA1D P25100 9/20 0.98
ADRA1B P35368 9/20 0.98
ADRB2 P07550 9/20 0.98
ADRB1 P08588 9/20 0.98
ADRB3 P13945 9/20 0.98
OPRL1 P41146 4/20 0.56
CHRM2 P08172 2/20 0.51
CHRM1 P11229 2/20 0.51
CHRM4 P08173 1/20 0.51
CHRM5 P08912 1/20 0.51
CHRM3 P20309 1/20 0.51
PLD1 Q13393 2/20 0.50
KCNH2 Q12809 2/20 0.50
OPRM1 P35372 2/20 0.50
OPRK1 P41145 2/20 0.50
YEATS4 O95619 1/20 0.50
MLLT3 P42568 1/20 0.50
MLLT1 Q03111 1/20 0.50
YEATS2 Q9ULM3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11430312 0.99 ADRA1D (1.00) ADRA1AADRA1DADRA1BADRB2ADRB1
Hydrochloric Acid SCHEMBL11432246 0.98 ADRA1D (0.98) ADRA1AADRA1DADRA1BADRB2ADRB1
SCHEMBL11428029 0.92 ADRA1A (0.83) ADRA1AADRA1DADRA1BADRB2ADRB1
SCHEMBL11443026 0.89 ADRA1D (0.98) ADRA1AADRA1DADRA1BADRB2ADRB1
SCHEMBL11441354 0.89 ADRA1D (0.79) ADRA1AADRA1DADRA1BADRB2ADRB1
Hydrochloric Acid SCHEMBL11427722 0.89 ADRA1D (1.00) ADRA1AADRA1DADRA1BADRB2ADRB1
Hydrochloric Acid SCHEMBL11439279 0.88 ADRA1D (0.85) ADRA1AADRA1DADRA1BADRB2ADRB1
SCHEMBL11427976 0.88 ADRA1D (0.77) ADRA1AADRA1DADRA1BADRB2ADRB1
Hydrochloric Acid SCHEMBL11032271 0.88 ADRA1A (0.80) ADRA1AADRA1DADRA1BADRB2ADRB1
SCHEMBL11437489 0.87 ADRA1D (0.98) ADRA1AADRA1DADRA1BADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4200755-A ADRENERGIC BLOCKING AGENTS, ANTISPASMODIC AGENTS, HYPOTENSIVE AGENTS RICHARDSON-MERRELL INC. (US) 1980-04-29 US claimed
US-4200755-A ADRENERGIC BLOCKING AGENTS, ANTISPASMODIC AGENTS, HYPOTENSIVE AGENTS RICHARDSON-MERRELL INC. (US) 1980-04-29 US disclosed