SCHEMBL1143744

SCHEMBL1143744

CO[C@@H](C=O)[C@@H](O)[C@@H](O)[C@H](O)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.39
TSHR P16473 2/20 0.36
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PGD P52209 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL645759 1.00 PDE4A (0.39) PDE4ATSHRSLC1A3SLC1A2SLC1A1
SCHEMBL570718 0.84 TSHR (0.33) TSHRSLC1A3SLC1A2SLC1A1
SCHEMBL5458333 0.84 TSHR (0.33) PDE4ATSHRSLC1A3SLC1A2SLC1A1
SCHEMBL7148889 0.84 TSHR (0.33) TSHRSLC1A3SLC1A2SLC1A1
SCHEMBL23923262 0.80 PDE4A (0.36) PDE4ATSHRCYP2C9ALDH1A1
SCHEMBL1037497 0.80 PDE4A (0.36) PDE4ATSHRCYP2C9ALDH1A1
SCHEMBL1950299 0.80 PDE4A (0.36) PDE4ATSHRCYP2C9ALDH1A1
SCHEMBL6258700 0.79 PDE4A (0.39) PDE4ATSHRCYP2C9ALDH1A1
SCHEMBL10885691 0.79 PDE4A (0.39) PDE4ATSHRCYP2C9ALDH1A1
SCHEMBL23925241 0.79 PDE4A (0.39) PDE4ATSHRCYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2797942-B1 COMPOSITION OF NOVEL CARBOHYDRATE DRUG FOR TREATMENT OF HUMAN DISEASES GALECTIN THERAPEUTICS INC (US) 2018-10-31 EP claimed
EP-2906227-B1 GALACTOSE-PRONGED CARBOHYDRATE COMPOUNDS FOR THE TREATMENT OF DIABETIC NEPHROPATHY AND ASSOCIATED DISORDERS GALECTIN THERAPEUTICS INC (US) 2018-10-03 EP claimed
WO-2006104503-A1 STRESS TOLERANT TRANSGENIC PLANTS OVER-EXPRESSING GENES OF ASCORBIC ACID SYNTHESIS-CELL WALL VIRGINIA TECH INTELLECTUAL PROPERTIES, INC. (US) 2006-10-05 WO claimed
EP-4044822-B1 CHOCOLATE PRODUCTS, INGREDIENTS, PROCESSES AND USES NESTLE SA (CH) 2024-05-15 EP disclosed
US-20240099326-A1 CHOCOLATE PRODUCTS, INGREDIENTS, PROCESSES AND USES SOCIETE DES PRODUITS NESTLE S.A. (CH) 2024-03-28 US disclosed
CN-116670296-A Method for producing sugar products and fermentation products 维尔萨利斯股份公司 2023-08-29 CN disclosed
CN-107406862-B Process for enzymatic hydrolysis of lignocellulosic material and fermentation of sugars 帝斯曼知识产权资产管理有限公司 2022-08-09 CN disclosed
US-20220225632-A1 CHOCOLATE PRODUCTS, INGREDIENTS, PROCESSES AND USES SOCIETE DES PRODUITS NESTLE S.A. (CH) 2022-07-21 US disclosed
US-20220217988-A1 CHOCOLATE PRODUCTS, INGREDIENTS, PROCESSES AND USES NESTLE SA (CH) 2022-07-14 US disclosed
US-11369122-B2 Chocolate products, ingredients, processes and uses SOCIETE DES PRODUITS NESTLE S.A. (CH) 2022-06-28 US disclosed
CN-107075533-B Process for enzymatic hydrolysis of lignocellulosic material and fermentation of sugars 帝斯曼知识产权资产管理有限公司 2021-11-02 CN disclosed
US-6177256-B1 VACCINE DIRECTED AGAINST TUMOR CELLS EXPRESSING MUCIN; CONJUGATE OF HUMAN MUCIN POLYPEPTIDE OR VARIABLE NUMBER OF TANDEM REPEATS AND OXIDIZED MANNAN IN A PHARMACEUTICALLY ACCEPTABLE CARRIER; ANTICANCER AGENTS AGAINST BREAST CANCER AUSTIN RESEARCH INSTITUTE (AU) 2001-01-23 US disclosed
EP-1027063-A1 MANNOSE RECEPTOR BEARING CELL LINE AND ANTIGEN COMPOSITION THE AUSTIN RESEARCH INSTITUTE (AU) 2000-08-16 EP disclosed
US-5989552-A Antigen carbohydrate compounds and their use in immunotherapy AUSTIN RESEARCH INSTITUTE (AU) 1999-11-23 US disclosed
US-5985593-A DETERMINATION OF MICROORGANISM CONTAINING MYCOLIC ACID IN EXTERIOR MEMBRANE; ENZYME LYSIS INTEGRATED RESEARCH TECHNOLOGY, L.L.C. (US) 1999-11-16 US disclosed
WO-1999016455-A1 MANNOSE RECEPTOR BEARING CELL LINE AND ANTIGEN COMPOSITION THE AUSTIN RESEARCH INSTITUTE (US) 1999-04-08 WO disclosed
WO-1995018145-A1 CONJUGATES OF HUMAN MUCIN AND A CARBOHYDRATE POLYMER AND THEIR USE IN CANCER TREATMENT ILEXUS PTY LTD (AU) 1995-07-06 WO disclosed
EP-0659768-A2 Antigen-carbohydrate conjugates and their use in immunotherapy ILEXUS PTY LTD (AU) 1995-06-28 EP disclosed
US-4617276-A SUBTRACTING THE DETERMINED AMOUNTS OF PROTEIN, LIPID, ASH AND NEUTRAL DETERGENT FIBER AGWAY INC. (US) 1986-10-14 US disclosed
US-4615891-A Method of formulating dairy cow rations based on carbohydrate regulation AGWAY INC. (US) 1986-10-07 US disclosed