SCHEMBL11440641

SCHEMBL11440641

NC(=O)NC(=O)c1c(Cl)cccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.53
TYK2 P29597 3/20 0.53
JAK1 P23458 3/20 0.53
CYP3A4 P08684 1/20 0.53
KMT2A Q03164 1/20 0.51
ALDH1A1 P00352 3/20 0.50
MAPT P10636 2/20 0.50
CYP1A2 P05177 1/20 0.50
SCN5A Q14524 1/20 0.49
SCN2A Q99250 1/20 0.49
PPIA P62937 1/20 0.49
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
TAS1R2 Q8TE23 1/20 0.49
HPGD P15428 1/20 0.49
GAA P10253 2/20 0.45
KDM4E B2RXH2 1/20 0.45
APAF1 O14727 1/20 0.45
TDP2 O95551 1/20 0.45
NSD2 O96028 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11499405 0.87 GAA (0.59) JAK2TYK2JAK1KMT2AMAPT
SCHEMBL8668403 0.84 MAPT (0.47) JAK2TYK2JAK1CYP3A4KMT2A
Hydrochloric Acid SCHEMBL7942179 0.82 MAPT (0.46) JAK2TYK2JAK1CYP3A4KMT2A
SCHEMBL16059203 0.79 JAK2 (0.57) JAK2JAK1KMT2AALDH1A1CYP1A2
SCHEMBL5467789 0.79 KDM4E (0.65) JAK2TYK2JAK1CYP3A4KMT2A
SCHEMBL4377125 0.78 ALDH1A1 (0.56) JAK2TYK2JAK1CYP3A4KMT2A
SCHEMBL9118696 0.78 POLB (0.64) JAK2TYK2KMT2AALDH1A1CYP1A2
SCHEMBL20387809 0.76 ALDH1A1 (0.50) JAK2TYK2JAK1CYP3A4ALDH1A1
Urea SCHEMBL10392049 0.76 KMT2A (0.56) JAK2TYK2JAK1CYP3A4KMT2A
SCHEMBL11005407 0.76 ALDH1A1 (0.56) JAK2TYK2JAK1CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0018144-A1 A process for the preparation of substituted 2-aminopyrazines ELI LILLY AND COMPANY (US) 1980-10-29 EP disclosed
US-4211870-A FROM AMINOACETONITRILE AND A PHENYL A-HALO OXIME ELI LILLY AND COMPANY (US) 1980-07-08 US disclosed
US-4164581-A 1-(2,6-Dichlorobenzoyl)-3-(4-trifluoromethyl-2-thiazolyl)urea and use as insecticide GULF OIL CORPORATION (US) 1979-08-14 US disclosed