SCHEMBL1144444

SCHEMBL1144444

NNc1ccc(S(N)(=O)=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 1.00
CA1 P00915 15/20 1.00
CA9 Q16790 14/20 1.00
CA12 O43570 13/20 1.00
CA6 P23280 4/20 1.00
CA5A P35218 4/20 1.00
CA7 P43166 4/20 1.00
CA5B Q9Y2D0 4/20 1.00
CA4 P22748 3/20 1.00
CA14 Q9ULX7 3/20 1.00
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
CA13 Q8N1Q1 2/20 0.54
USP2 O75604 1/20 0.54
TSHR P16473 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
AGO2 Q9UKV8 1/20 0.54
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrazine SCHEMBL7570110 0.98 CA2 (0.95) CA2CA1CA9CA12CA6
Hydrochloric Acid SCHEMBL6696969 0.98 CA2 (0.95) CA2CA1CA9CA12CA6
Hydrochloric Acid SCHEMBL981171 0.98 CA2 (0.95) CA2CA1CA9CA12CA6
Hydrochloric Acid SCHEMBL27493662 0.95 CA2 (0.91) CA2CA1CA9CA12CA6
Hypochlorous Acid SCHEMBL5859040 0.93 CA2 (0.87) CA2CA1CA9CA12CA6
SCHEMBL4640918 0.82 ALDH1A1 (0.79) CA2CA1CA9CA12CA6
SCHEMBL28102126 0.82 CA2 (0.70) CA2CA1CA9CA12CA6
SCHEMBL28107398 0.82 SOS1 (0.70) CA2CA1CA9CA12CA6
SCHEMBL22001051 0.81 CA2 (0.68) CA2CA1CA9CA12CA6
SCHEMBL202948 0.81 CA2 (0.81) CA2CA1CA9CA12CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 358 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114478493-B Traceable 5-aminosalicylic acid derivative and preparation and application thereof 中国科学院兰州化学物理研究所 2024-04-02 CN claimed
CN-115784947-A COX-II enzyme inhibitor celecoxib intermediate and synthesis method thereof 药大制药有限公司 2023-03-14 CN claimed
CN-110526868-B Preparation method of celecoxib 迪嘉药业集团有限公司 2022-03-18 CN claimed
CN-112986410-A Method for detecting arylamine and aromatic hydrazine gene toxic impurities in celecoxib 南京亿华药业有限公司 2021-06-18 CN claimed
CN-111423375-A Preparation method of COX-2 specific cyclooxygenase inhibitor 云南大学 2020-07-17 CN claimed
CN-111217753-A Preparation method of celecoxib 农永强 2020-06-02 CN claimed
CN-110698404-A Preparation method of high-purity celecoxib 安徽恒星制药有限公司 2020-01-17 CN claimed
CN-110526868-A A kind of preparation method of celecoxib WEIHAI DISU PHARMACEUTICAL CO LTD 2019-12-03 CN claimed
CN-109689627-A Pyrazolyl quinoline compound and preparation method thereof and medical component 高雄医学大学 2019-04-26 CN claimed
CN-106480439-A A kind of chemical nickel plating palldium alloy crosses liquid and its application 江苏澳光电子有限公司 2017-03-08 CN claimed
EP-1191931-A4 1-(4-SULFAMYLARYL)-3-SUBSTITUTED-5-ARYL-2-PYRAZOLINES AS INHIBITORS OF CYCLOOXYGENASE-2 UNIV TEMPLE (US) 2002-11-27 EP claimed
EP-0828717-B1 METHOD OF PREPARING 3-HALOALKYL-1H-PYRAZOLES SEARLE & CO (US) 2002-09-04 EP claimed
US-6376519-B1 ANTIINFLAMMATORY AGENTS, ANTICANCER AGENTS TEMPLE UNIVERSITY-OF THE COMMONWEALTH OF HIGHER EDUCATION 2002-04-23 US claimed
EP-1191931-A1 1-(4-SULFAMYLARYL)-3-SUBSTITUTED-5-ARYL-2-PYRAZOLINES AS INHIBITORS OF CYCLOOXYGENASE-2 Temple University of the Commonwealth System of Higher Education (US) 2002-04-03 EP claimed
WO-2000076503-A1 1-(4-SULFAMYLARYL)-3-SUBSTITUTED-5-ARYL-2-PYRAZOLINES AS INHIBITORS OF CYCLOOXYGENASE-2 TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2000-12-21 WO claimed
US-5910597-A Process for preparing 3-haloalkyl-1H-pyrazoles G.D. SEARLE & CO. (US) 1999-06-08 US claimed
US-5892053-A Process for preparing 3-haloalkyl-1H-pyrazoles G. D. SEARLE & CO. (US) 1999-04-06 US claimed
CN-1190960-A Method of preparing 3-haloalkyl-1H-pyrazoles SEARLE & CO (US) 1998-08-19 CN claimed
EP-0828717-A1 METHOD OF PREPARING 3-HALOALKYL-1H-PYRAZOLES G.D. SEARLE & CO. (US) 1998-03-18 EP claimed
WO-1996037476-A1 METHOD OF PREPARING 3-HALOALKYL-1H-PYRAZOLES G.D. SEARLE & CO. (US) 1996-11-28 WO claimed