SCHEMBL11449581

SCHEMBL11449581

COC(=O)C1CCC(OC)CN1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.36
CHRNA4 P43681 2/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA7 P36544 1/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CTSC P53634 1/20 0.33
KMT2A Q03164 1/20 0.33
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15248182 1.00 CHRNB2 (0.36) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL11449583 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL6199839 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL13403384 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL10151348 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL5605655 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL7021231 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL3834619 0.82 CTSC (0.42) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL11449155 0.82 HRH3 (0.31)
Hydrochloric Acid SCHEMBL7321361 0.81 CTSC (0.41) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4221912-A Dithio derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-09-09 US disclosed
US-4217458-A Acylmercaptoacyl derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-08-12 US disclosed
US-4198515-A Mercaptoacyl derivatives of 4,5-dihydro-1H-pyrrole-2-carboxylic acids and 1,4,5,6-tetrahydropyridine-2-carboxylic acids E. R. SQUIBB & SONS, INC. (US) 1980-04-15 US disclosed