Fosazepam

Fosazepam

SCHEMBL114556

CP(C)(=O)CN1C(=O)CN=C(c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.69
NR1I2 O75469 1/20 0.69
ADORA3 P0DMS8 1/20 0.69
OPRM1 P35372 1/20 0.69
TP53 P04637 5/20 0.69
GABRA1 P14867 3/20 0.67
GABRA5 P31644 3/20 0.67
GABRA3 P34903 3/20 0.67
GABRA2 P47869 3/20 0.67
GABRB2 P47870 3/20 0.67
GABRG2 P18507 2/20 0.67
GABRB3 P28472 2/20 0.67
GABRP O00591 1/20 0.67
GABRD O14764 1/20 0.67
CACNA1F O60840 1/20 0.67
ALB P02768 1/20 0.67
GABRB1 P18505 1/20 0.67
AKR1C3 P42330 1/20 0.67
GABRA4 P48169 1/20 0.67
AKR1C2 P52895 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5355886 0.87 OPRK1 (0.73) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL11855695 0.86 OPRK1 (0.69) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL5361417 0.85 OPRK1 (0.72) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL3579580 0.85 OPRK1 (0.73) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL5349082 0.85 TP53 (0.84) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL16777701 0.83 NPSR1 (0.72) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL11576383 0.83 OPRK1 (0.68) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL9040148 0.83 OPRK1 (0.71) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL9039066 0.83 CYP1A2 (0.75) OPRK1NR1I2ADORA3OPRM1TP53
SCHEMBL11577195 0.83 OPRK1 (0.65) OPRK1NR1I2ADORA3OPRM1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2518 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024150170-A1 PIROMELATINE FOR TREATING PARASOMNIAS ASSOCIATED WITH LOSS OF REM SLEEP ATONIA NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2024-07-18 WO claimed
US-20240238250-A1 METHOD OF USING PIROMELATINE FOR TREATING PARASOMNIAS ASSOCIATED WITH LOSS OF REM SLEEP ATONIA NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2024-07-18 US claimed
US-10689373-B2 1,2-substituted cyclopentanes as orexin receptor antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-06-23 US claimed
US-20190275048-A1 METHOD OF TREATING INSOMNIA ROSENBERG LEON I (US) 2019-09-12 US claimed
US-20180282309-A1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-10-04 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8735383-B2 Glycine transporter-1 inhibitors AMGEN INC. (US) 2014-05-27 US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20120195985-A1 GLYCINE TRANSPORTER-1 INHIBITORS AMGEN INC. (US) 2012-08-02 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
EP-1599199-A2 METHODS FOR TREATING JOINT PAIN OR IMPROVING SLEEP USING AN ESTROGEN AGONIST/ANTAGONIST Pfizer Products Inc. (US) 2005-11-30 EP claimed
WO-2004064832-A2 METHODS FOR TREATING JOINT PAIN OR IMPROVING SLEEP USING AN ESTROGEN AGONIST/ANTAGONIST PFIZER PRODUCTS INC. (US) 2004-08-05 WO claimed
US-20040152713-A1 Methods for treating joint pain or improving sleep using an estrogen agonist/antagonist PFIZER INC. 2004-08-05 US claimed
JP-2000511885-A 2000-09-12 JP claimed
EP-0900086-A4 ENHANCEMENT OF SLEEP WITH A GROWTH HORMONE SECRETAGOGUE MERCK & CO INC (US) 2000-01-12 EP claimed
EP-0900086-A1 ENHANCEMENT OF SLEEP WITH A GROWTH HORMONE SECRETAGOGUE Merck & Co., Inc. (US) 1999-03-10 EP claimed
WO-1997041879-A1 ENHANCEMENT OF SLEEP WITH A GROWTH HORMONE SECRETAGOGUE MERCK & CO., INC. (US) 1997-11-13 WO claimed
US-4557934-A ALONG WITH A DIOL PYRROLIDONE OR AN AZACYCLOPENTAN-2-ONE THE PROCTER & GAMBLE COMPANY (US) 1985-12-10 US claimed