SCHEMBL11455692

SCHEMBL11455692

COc1ccc2c(c1)CCN(CC1CCCC1)CC2

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.64
HRH1 P35367 2/20 0.58
CYP2D6 P10635 1/20 0.57
SIGMAR1 Q99720 2/20 0.54
HTR1A P08908 1/20 0.54
OPRM1 P35372 3/20 0.52
OPRL1 P41146 2/20 0.52
OPRK1 P41145 1/20 0.52
DRD2 P14416 4/20 0.51
DRD1 P21728 4/20 0.51
DRD5 P21918 4/20 0.51
DRD3 P35462 4/20 0.51
DRD4 P21917 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11459467 0.97 HRH3 (0.60) HRH3HRH1CYP2D6SIGMAR1HTR1A
SCHEMBL11466219 0.94 HRH3 (0.64) HRH3HRH1CYP2D6SIGMAR1HTR1A
SCHEMBL2567353 0.91 HRH3 (0.67) HRH3HRH1CYP2D6SIGMAR1HTR1A
SCHEMBL12950793 0.89 HRH3 (0.62) HRH3HRH1CYP2D6SIGMAR1HTR1A
SCHEMBL5904101 0.81 SIGMAR1 (0.71) HRH3HRH1SIGMAR1HTR1AOPRM1
SCHEMBL29438692 0.80 HRH3 (0.53) HRH3HRH1CYP2D6SIGMAR1HTR1A
SCHEMBL4923590 0.79 HRH3 (0.77) HRH3HRH1CYP2D6
Hydrochloric Acid SCHEMBL4622628 0.79 SIGMAR1 (0.68) HRH3HRH1SIGMAR1HTR1A
SCHEMBL11457338 0.79 DRD1 (0.60) HRH3DRD2DRD1DRD5DRD3
SCHEMBL6071227 0.78 HRH3 (1.00) HRH3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4233217-A USED AS ANALGESICS, NARCOTIC ANTAGONISTS, AND ANTIHISTAMINES PENNWALT CORPORATION (US) 1980-11-11 US disclosed
US-4210749-A USED AS ANALGESICS, NARCOTIC ANTAGONISTS PENNWALT CORPORATION (US) 1980-07-01 US disclosed