SCHEMBL29438692

SCHEMBL29438692

COc1ccc2c(c1)CCN(CC1CCOCC1)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.53
THRB P10828 1/20 0.47
DRD1 P21728 2/20 0.47
DRD5 P21918 2/20 0.47
SIGMAR1 Q99720 3/20 0.47
PRMT5 O14744 1/20 0.47
HRH1 P35367 2/20 0.46
CYP2D6 P10635 1/20 0.46
DRD3 P35462 2/20 0.46
DRD2 P14416 1/20 0.46
KDM4E B2RXH2 1/20 0.44
HTR1A P08908 2/20 0.44
CHRM2 P08172 1/20 0.44
CHRM3 P20309 1/20 0.44
DRD4 P21917 1/20 0.44
ADRA1D P25100 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
HTR2B P41595 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12950793 0.88 HRH3 (0.62) HRH3THRBDRD1DRD5SIGMAR1
SCHEMBL31534242 0.83 ABCB1 (0.52) KDM4E
SCHEMBL11466219 0.83 HRH3 (0.64) HRH3DRD1DRD5SIGMAR1HRH1
SCHEMBL2567353 0.82 HRH3 (0.67) HRH3THRBDRD1DRD5SIGMAR1
SCHEMBL30068748 0.81 THRB (0.46) HRH3THRBSIGMAR1HRH1DRD3
SCHEMBL30845461 0.81 DRD2 (0.47) HRH3DRD1DRD5SIGMAR1PRMT5
SCHEMBL11455692 0.80 HRH3 (0.64) HRH3DRD1DRD5SIGMAR1HRH1
SCHEMBL11459467 0.80 HRH3 (0.60) HRH3DRD1DRD5SIGMAR1HRH1
SCHEMBL12719849 0.80 PKM (0.55) HRH3THRBCYP2D6
Hydrochloric Acid SCHEMBL1626954 0.79 PKM (0.54) HRH3THRBCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114195764-A Compound as thyroid hormone beta receptor agonist and application thereof 广东东阳光药业有限公司 2022-03-18 CN disclosed