SCHEMBL11458609

SCHEMBL11458609

C=CCC1(C(CC)C(=O)O)CCCc2ccc(OC)cc21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.40
POLA1 P09884 2/20 0.39
AKR1C3 P42330 3/20 0.36
AKR1C2 P52895 3/20 0.36
CXCR5 P32302 1/20 0.36
AKR1C1 Q04828 1/20 0.36
PTGS1 P23219 1/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP3A4 P08684 1/20 0.35
KIF11 P52732 1/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11457214 0.79 AKR1C3 (0.39) POLA1AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL6583622 0.78 POLA1 (0.46) SIGMAR1POLA1CXCR5CYP2C19CYP2C9
SCHEMBL28735232 0.73 SIGMAR1 (0.45) SIGMAR1POLA1CYP2C19CYP2C9TSHR
SCHEMBL11458608 0.72 OPRM1 (0.39) SIGMAR1POLA1CYP2C19CYP2C9TSHR
SCHEMBL11459393 0.71 AKR1C3 (0.46) POLA1AKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL30067572 0.70 KDM1A (0.41) KDM1A
SCHEMBL16388051 0.70 KDM1A (0.45) SIGMAR1POLA1CYP2C19CYP2C9TSHR
SCHEMBL18487244 0.69 POLA1 (0.46) SIGMAR1POLA1AKR1C3AKR1C2PTGS1
SCHEMBL6580889 0.68 POLA1 (0.55) SIGMAR1POLA1CYP2C19CYP2C9TSHR
SCHEMBL5396757 0.68 POLA1 (0.52) SIGMAR1POLA1CXCR5KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4234731-A BROMINATION AND SALT FORMATION OF BENZ(E)INDOLINES; HYDROLYSIS WITH A BICARBONATE; RING EXPANSION AND REARRANGEMENT BRISTOL-MYERS COMPANY (US) 1980-11-18 US disclosed
US-4150032-A ANALGESIC, ANTITUSSIVE BRISTOL-MYERS COMPANY (US) 1979-04-17 US disclosed