SCHEMBL1146008

SCHEMBL1146008

COC1CCCS1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12678305 0.92
SCHEMBL15953782 0.79
SCHEMBL79191 0.77 NOS2 (0.33)
SCHEMBL5648243 0.77 NOS2 (0.33)
SCHEMBL15328487 0.72
SCHEMBL1146005 0.72
SCHEMBL4609280 0.72
SCHEMBL20601576 0.72
SCHEMBL10823486 0.72
SCHEMBL78700 0.70 KDM4E (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073373-A Method for asymmetric synthesis of (R) -5' -methoxy labdanin 广东嘉博制药有限公司 2022-09-20 CN disclosed
CN-111004179-B Resolution method of 5' -methoxylapatin 武汉大安制药有限公司 2021-03-09 CN disclosed
CN-111004179-A Resolution method of 5' -methoxylapatin 武汉大安制药有限公司 2020-04-14 CN disclosed
CN-104334717-B The dewaxing buffer solution of containing water-soluble organic solvent and its using method 理查艾伦科学公司 2017-03-15 CN disclosed
CN-104380107-B The method preparing biology sensor 诺威奥森斯有限公司 2016-11-02 CN disclosed
CN-102782927-B Nonaqueous electrolyte solution, electrochemical element using same, and 1,2-dioxypropane compound used in same UBE INDUSTRIES 2015-07-15 CN disclosed
CN-104380107-A Process for making biosensor NOVIOSENSE B V 2015-02-25 CN disclosed
CN-104334717-A Dewaxing buffer containing a water-soluble organic solvent and methods of use thereof RICHARD ALLAN SCIENT COMPANY 2015-02-04 CN disclosed
US-7888374-B2 Inhibitors of c-jun N-terminal kinases ABBOTT LABORATORIES (US) 2011-02-15 US disclosed
WO-2006083673-A2 PYRIDINE DERIVATIVES USEFUL AS INHIBITORS OF C-JUN N-TERMINAL KINASES ABBOTT LABORATORIES (US) 2006-08-10 WO disclosed
US-20060173050-A1 Inhibitors of c-Jun N-terminal kinases ABBVIE INC. 2006-08-03 US disclosed
US-20050171132-A1 Diaminopyrimidine derivatives as selective growth hormone secrectgogue receptor (GHS-R) antagonists XIN ZHILI (US) 2005-08-04 US disclosed
US-20050171131-A1 Diaminopyrimidine derivatives as growth hormone secrectgogue receptor (GHS-R) antagonists KOSOGOF CHRISTI (US) 2005-08-04 US disclosed
WO-2005030734-A1 DIAMINOPYRIMIDINE DERIVATIVES AS SELECTIVE GROWTH HORMONE SECRECTGOGUE RECEPTOR (GHS-R) ANTAGONISTS ABBOTT LABORATORIES (US) 2005-04-07 WO disclosed
US-20050070712-A1 Pyrimidine derivatives as ghrelin receptor modulators ABBOTT LABORATORIES 2005-03-31 US disclosed
US-3970679-A Process for the production of organotin halides in sulphones as reaction medium CIBA-GEIGY CORPORATION (US) 1976-07-20 US disclosed