SCHEMBL11468997

SCHEMBL11468997

O=c1[nH]ccc(-c2ccncc2)c1CO

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.60
MAPK14 Q16539 2/20 0.44
GCGR P47871 1/20 0.44
GSK3B P49841 2/20 0.42
PDE3B Q13370 5/20 0.41
PDE3A Q14432 5/20 0.41
AURKB Q96GD4 2/20 0.41
INCENP Q9NQS7 2/20 0.41
JAK2 O60674 1/20 0.40
CCNC P24863 4/20 0.40
CDK8 P49336 4/20 0.40
PIK3CD O00329 1/20 0.40
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
HPGD P15428 2/20 0.38
PDE4A P27815 2/20 0.38
CYP2C19 P33261 2/20 0.38
BLM P54132 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12984897 0.84 PADI4 (0.49) MAPTGSK3BAURKBINCENPCYP2C19
SCHEMBL7511441 0.75 MAPT (0.58) MAPTMAPK14GCGRGSK3BPDE3B
SCHEMBL11449584 0.71 MAPT (0.58) MAPTMAPK14GCGRGSK3BPDE3B
SCHEMBL2100160 0.71 MAPT (0.58) MAPTMAPK14GCGRGSK3BPDE3B
Hydrochloric Acid SCHEMBL30730902 0.69 MAPT (0.56) MAPTMAPK14GCGRGSK3BPDE3B
SCHEMBL11291385 0.69 PDE3B (0.63) MAPTGSK3BPDE3BPDE3AAURKB
SCHEMBL17060505 0.68 DAO (0.34) MAPTAURKBINCENPKDM4ELMNA
SCHEMBL14912178 0.68 MAPT (0.54) MAPTMAPK14GCGRGSK3BJAK2
SCHEMBL14912198 0.67 MAPT (0.53) MAPTMAPK14GCGRGSK3BAURKB
SCHEMBL6535945 0.67 MAPT (0.56) MAPTPDE3BPDE3AJAK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4225601-A 3-Hydroxy or hydroxymethyl-5-(4-pyridinyl)2(1H)-pyridinones, useful as cardiotonic agents and their preparation STERLING DRUG INC. (US) 1980-09-30 US disclosed