SCHEMBL11479727

SCHEMBL11479727

O=C(O)CCCc1ccc(-n2ccnc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 7/20 1.00
CYP3A4 P08684 3/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
RXRA P19793 1/20 0.52
RXRB P28702 1/20 0.52
RXRG P48443 1/20 0.52
ADH5 P11766 1/20 0.52
BAZ2B Q9UIF8 1/20 0.51
ENPP2 Q13822 1/20 0.50
MKNK1 Q9BUB5 1/20 0.50
MKNK2 Q9HBH9 1/20 0.50
HDAC3 O15379 1/20 0.49
MAPK1 P28482 1/20 0.49
ADRA1A P35348 1/20 0.49
HDAC4 P56524 1/20 0.49
SLC6A3 Q01959 1/20 0.49
HDAC1 Q13547 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11475605 0.83 TBXAS1 (0.71) TBXAS1CYP3A4HDAC3MAPK1ADRA1A
SCHEMBL7434598 0.81 TBXAS1 (0.68) TBXAS1CYP3A4ADH5BAZ2BENPP2
SCHEMBL11484688 0.81 TBXAS1 (0.68) TBXAS1CYP3A4CYP2D6CYP2C9BAZ2B
SCHEMBL10762282 0.81 TBXAS1 (0.68) TBXAS1CYP3A4CYP2D6CYP2C9ADH5
SCHEMBL11449452 0.80 CYP2D6 (0.68) TBXAS1CYP3A4CYP2D6CYP2C9
SCHEMBL11477536 0.80 TBXAS1 (0.66) TBXAS1CYP3A4
SCHEMBL28108298 0.78 CYP3A4 (0.65) TBXAS1CYP3A4CYP2D6CYP2C9BAZ2B
Hydrochloric Acid SCHEMBL11477573 0.78 TBXAS1 (1.00) TBXAS1CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8392830 0.78 CYP3A4 (0.69) TBXAS1CYP3A4CYP2D6CYP2C9ADH5
SCHEMBL7275362 0.78 TBXAS1 (0.63) TBXAS1CYP3A4CYP2D6CYP2C9ADH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4226878-A ANTIINFLAMMATORY, HYPOTENSIVES, ANTIHISTAMINES KISSEI PHARMACEUTICAL CO., LTD. (JP) 1980-10-07 US disclosed