SCHEMBL11488183

SCHEMBL11488183

CC(CCBr)c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.39
FFAR1 O14842 1/20 0.37
DPP4 P27487 1/20 0.34
KCNH2 Q12809 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1543906 0.94 AOC3 (0.36) AOC3
SCHEMBL3756197 0.82 CACNA1B (0.35) AOC3
SCHEMBL13792137 0.82 ALDH1A1 (0.41) CYP17A1FFAR1
SCHEMBL11487942 0.81 CYP17A1 (0.48) CYP17A1FFAR1DPP4KCNH2DPP8
SCHEMBL27900218 0.81 CYP17A1 (0.39) CYP17A1FFAR1DPP4KCNH2DPP8
SCHEMBL11493405 0.81 TRPA1 (0.42) CYP17A1FFAR1DPP4KCNH2DPP8
SCHEMBL11487070 0.81 MAOB (0.46) CYP17A1FFAR1DPP4KCNH2DPP8
Hydrochloric Acid SCHEMBL11493325 0.79 MAOB (0.48) CYP17A1FFAR1DPP4KCNH2DPP8
SCHEMBL11493802 0.79 MAOB (0.42) CYP17A1FFAR1DPP4KCNH2DPP8
SCHEMBL11489248 0.79 CYP17A1 (0.39) CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4239759-A Morpholino containing compounds, compositions and use thereof MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-12-16 US disclosed
US-4110447-A Anti-inflammatory (halo-4-biphenylyl)-alkanolamines MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1978-08-29 US disclosed