SCHEMBL1149037

SCHEMBL1149037

Cc1nc2ccc(Oc3ccc(C(F)(F)F)cc3Cl)c(C(F)(F)F)c2c(O)c1C

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.37
PDE2A O00408 6/20 0.36
MRGPRX4 Q96LA9 6/20 0.36
PDE10A Q9Y233 2/20 0.35
MEN1 O00255 1/20 0.35
TTR P02766 1/20 0.35
PPOX P50336 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ESRRA P11474 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1149203 0.86 DHODH (0.35) FFAR1PDE2AMRGPRX4PDE10A
SCHEMBL1148866 0.83 FFAR1 (0.38) FFAR1MRGPRX4MEN1TTRPPOX
SCHEMBL1148825 0.79 FFAR1 (0.36) FFAR1PDE2AMRGPRX4MEN1TTR
SCHEMBL1148810 0.76 SLC6A4 (0.36) PDE2APDE10A
SCHEMBL14715540 0.75 PDE3B (0.31)
SCHEMBL10707742 0.71 FFAR1 (0.54) FFAR1PDE2AMRGPRX4MEN1TTR
SCHEMBL2823352 0.71 PDE2A (0.31) PDE2A
SCHEMBL7803868 0.69 AR (0.46) FFAR1PDE2AMRGPRX4MEN1TTR
SCHEMBL7803948 0.69 TTR (0.49) FFAR1PDE2AMRGPRX4MEN1TTR
SCHEMBL1148924 0.68 FFAR1 (0.37) FFAR1MRGPRX4MEN1TTRPPOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1780202-B1 QUINOLINE DERIVATIVE AND INSECTICIDE CONTAINING SAME AS ACTIVE CONSTITUENT MEIJI SEIKA PHARMA CO LTD (JP) 2013-02-27 EP disclosed
US-7880006-B2 4-Acetoxy-5-chloro-6-(4-chlorophenoxy)-2,3-dimethyl-quinoline, used as agricultural and horticultural insecticides MEIJI SEIKA KAISHA, LTD. (JP) 2011-02-01 US disclosed
US-20070203181-A1 Quinoline Derivatives And Insecticide Comprising Thereof As Active Ingredient MEIJI SEIKA KAISHA, LTD. (JP) 2007-08-30 US disclosed
EP-1780202-A1 QUINOLINE DERIVATIVE AND INSECTICIDE CONTAINING SAME AS ACTIVE CONSTITUENT MEIJI SEIKA KAISHA LTD. (JP) 2007-05-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070203181-A1 Quinoline Derivatives And Insecticide Comprising Thereof As Active Ingredient DDT, ACHE, NQO1 FFAR1 2742/4885PDE2A 263/4885MRGPRX4 3431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.