SCHEMBL11501501

SCHEMBL11501501

CC(=O)NC(C#N)(NC(C)=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HDAC9 Q9UKV0 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
MAPT P10636 3/20 0.41
KMT2A Q03164 2/20 0.41
KCNN4 O15554 1/20 0.40
NAPRT Q6XQN6 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ALDH1A1 P00352 2/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C1 Q04828 1/20 0.38
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27803999 0.80 HDAC3 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7220861 0.76 ALDH1A1 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL31358110 0.74 KCNN4 (0.47) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3322720 0.74 MAPT (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8226385 0.74 KCNN4 (0.50) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL27346817 0.73 HDAC3 (0.46) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL13881112 0.72 KCNN4 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL2283304 0.72 SSTR4 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4566798 0.72 MAPT (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL15881583 0.71 KCNN4 (0.44) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003461-B1 AMINOALCOHOL DERIVATIVES OF ORTHO-HYDROXY-METHYL CINNAMATE, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1981-04-29 EP disclosed
EP-0003461-A1 Aminoalcohol derivatives of ortho-hydroxy-methyl cinnamate, process for their preparation and medicines containing them LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1979-08-08 EP disclosed