SCHEMBL11510985

SCHEMBL11510985

COC(=O)[C@@H](NC(=O)c1ccc(Oc2ccc(Cl)cc2)cc1)C(C)C

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.57
TAS1R1 Q7RTX1 1/20 0.57
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
NPSR1 Q6W5P4 2/20 0.49
ALDH1A1 P00352 1/20 0.48
UTS2R Q9UKP6 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MMP1 P03956 1/20 0.47
HTT P42858 2/20 0.47
TRPA1 O75762 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CCR1 P32246 2/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
PTGS2 P35354 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11508615 0.89 TAS1R3 (0.59) TAS1R3TAS1R1LMNANPSR1ALDH1A1
SCHEMBL11508045 0.87 TAS1R3 (0.58) TAS1R3TAS1R1LMNAMAPK1NPSR1
SCHEMBL11509367 0.87 TAS1R3 (0.62) TAS1R3TAS1R1LMNANPSR1ALDH1A1
SCHEMBL26814843 0.81 TAS1R3 (0.64) TAS1R3TAS1R1LMNAMAPK1NPSR1
SCHEMBL16234929 0.81 TRPA1 (0.56) TAS1R3TAS1R1LMNAMAPK1NPSR1
SCHEMBL26820886 0.79 TAS1R3 (0.70) TAS1R3TAS1R1LMNANPSR1ALDH1A1
SCHEMBL31595936 0.78 TAS1R3 (0.64) TAS1R3TAS1R1LMNANPSR1ALDH1A1
SCHEMBL16235094 0.77 TRPA1 (0.66) LMNAMAPK1ALDH1A1HTTTRPA1
SCHEMBL27564141 0.77 HTT (0.56) LMNAMAPK1ALDH1A1SMN1; SMN2HTT
SCHEMBL11509188 0.77 NPSR1 (0.66) TAS1R3TAS1R1LMNANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4161529-A Phenoxy phenyl pyrrolidine compounds, compositions and methods of use SCIENCE UNION ET CIE, SOCIETE FRANCAISE DE RECHERCHE MEDICALE (FR) 1979-07-17 US disclosed