SCHEMBL11517376

SCHEMBL11517376

COc1ccc2c(c1)c(CCN1CCN(C)CC1)c(C)n2C(=O)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.68
CNR1 P21554 4/20 0.68
TSHR P16473 2/20 0.67
LMNA P02545 2/20 0.67
CYP1A2 P05177 2/20 0.67
CYP2D6 P10635 2/20 0.67
CYP2C9 P11712 2/20 0.67
HIF1A Q16665 2/20 0.67
NPSR1 Q6W5P4 2/20 0.67
NFKB1 P19838 1/20 0.67
PLA2G2A P14555 1/20 0.65
AKR1C3 P42330 7/20 0.60
AKR1C2 P52895 5/20 0.60
PTGS1 P23219 3/20 0.59
MTOR P42345 2/20 0.59
TP53 P04637 1/20 0.59
CYP3A4 P08684 1/20 0.59
HPGD P15428 1/20 0.59
ALOX15 P16050 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11522517 0.85 CNR2 (0.59) CNR2CNR1TSHRLMNACYP1A2
SCHEMBL11518423 0.84 TSHR (0.60) CNR2CNR1TSHRLMNACYP1A2
SCHEMBL11520081 0.84 PTGS1 (0.80) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL11522535 0.83 LMNA (0.76) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL11518964 0.82 LMNA (0.62) CNR2CNR1TSHRLMNACYP1A2
SCHEMBL12949361 0.82 LMNA (0.80) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL1082631 0.81 HIF1A (1.00) TSHRLMNACYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL11517674 0.80 LMNA (0.59) CNR2CNR1TSHRLMNACYP1A2
Hydrochloric Acid SCHEMBL8646699 0.80 HIF1A (0.98) TSHRLMNACYP1A2CYP2D6CYP2C9
SCHEMBL23391007 0.79 LMNA (0.83) CNR2TSHRLMNACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160862-A ANTIINFLAMMATORY STERLING DRUG INC. (US) 1979-07-10 US disclosed
US-4021431-A ANTIINFLAMMATORY AGENTS STERLING DRUG INC. (US) 1977-05-03 US disclosed