SCHEMBL11517481

SCHEMBL11517481

COC(=O)C(C)c1cc2c(c(OC(C)=O)c1)C(=O)c1ccccc1CC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.55
ALDH1A1 P00352 5/20 0.42
MAPT P10636 4/20 0.42
MEN1 O00255 2/20 0.42
PKM P14618 2/20 0.42
KMT2A Q03164 2/20 0.42
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
PGAM1 P18669 1/20 0.38
PGR P06401 2/20 0.38
TTR P02766 2/20 0.38
CES1 P23141 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HPGD P15428 2/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 2/20 0.36
ABCC4 O15439 1/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11519977 0.90 AKR1B1 (0.58) AKR1B1ALDH1A1MAPTMEN1KMT2A
SCHEMBL11517611 0.89 AKR1B1 (0.53) AKR1B1ALDH1A1MAPTMEN1PKM
SCHEMBL11519465 0.89 AKR1B1 (0.69) AKR1B1ALDH1A1MAPTMEN1PKM
SCHEMBL11520526 0.86 AKR1B1 (0.54) AKR1B1ALDH1A1MAPTPTGS1PTGS2
SCHEMBL11519573 0.84 AKR1B1 (0.76) AKR1B1ALDH1A1MAPTMEN1PKM
SCHEMBL11517083 0.80 AKR1B1 (0.72) AKR1B1ALDH1A1MAPTMEN1PKM
SCHEMBL11843846 0.79 AKR1B1 (0.51) AKR1B1PTGS1PTGS2CES1L3MBTL1
SCHEMBL11517540 0.78 AKR1B1 (0.67) AKR1B1ALDH1A1MAPTMEN1PKM
SCHEMBL11520301 0.75 AKR1B1 (0.68) AKR1B1MAPTMEN1PKMKMT2A
SCHEMBL11518749 0.74 AKR1B1 (0.44) AKR1B1ALDH1A1MAPTMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172949-A 2,4-Disubstituted-5-oxo-5H-dibenzo[a,d]cycloheptenes SYNTEX (U.S.A.) INC. (US) 1979-10-30 US disclosed