SCHEMBL11519977

SCHEMBL11519977

COC(=O)C(C)c1cc2c(c(OC)c1)C(=O)c1ccccc1CC2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.58
POLB P06746 1/20 0.42
MAOA P21397 1/20 0.42
MIF P14174 1/20 0.42
MAPT P10636 9/20 0.42
ALDH1A1 P00352 7/20 0.42
SMN1; SMN2 Q16637 6/20 0.42
LMNA P02545 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HTT P42858 2/20 0.42
CASP3 P42574 2/20 0.42
SENP8 Q96LD8 2/20 0.42
SENP7 Q9BQF6 2/20 0.42
SENP6 Q9GZR1 2/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 2/20 0.41
USP2 O75604 1/20 0.41
DUSP3 P51452 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11517481 0.90 AKR1B1 (0.55) AKR1B1POLBMAOAMIFMAPT
SCHEMBL11517083 0.89 AKR1B1 (0.72) AKR1B1POLBMAOAMIFMAPT
SCHEMBL11520526 0.89 AKR1B1 (0.54) AKR1B1MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL11517611 0.88 AKR1B1 (0.53) AKR1B1POLBMAOAMIFMAPT
SCHEMBL11519573 0.87 AKR1B1 (0.76) AKR1B1POLBMAOAMIFMAPT
SCHEMBL11843846 0.82 AKR1B1 (0.51) AKR1B1TDP1RAB9APTGS1PTGS2
SCHEMBL11519465 0.78 AKR1B1 (0.69) AKR1B1MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL11523218 0.78 MAPT (0.49) AKR1B1POLBMAOAMIFMAPT
SCHEMBL11520301 0.77 AKR1B1 (0.68) AKR1B1MAPTSMN1; SMN2LMNAMEN1
SCHEMBL11517807 0.77 SRD5A1 (0.51) AKR1B1POLBMAOAMIFMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172949-A 2,4-Disubstituted-5-oxo-5H-dibenzo[a,d]cycloheptenes SYNTEX (U.S.A.) INC. (US) 1979-10-30 US disclosed