SCHEMBL11517540

SCHEMBL11517540

CCC(=O)Oc1cc(C(C)C(=O)O)cc2c1C(=O)c1ccccc1CC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.67
PTGS2 P35354 2/20 0.39
OPRK1 P41145 1/20 0.39
PDE4D Q08499 1/20 0.39
AKR1C3 P42330 3/20 0.38
AKR1C2 P52895 3/20 0.38
KMT2A Q03164 3/20 0.38
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
DRD1 P21728 2/20 0.38
MEN1 O00255 2/20 0.38
PKM P14618 2/20 0.38
LMNA P02545 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPC1 O15118 1/20 0.38
PGR P06401 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
NFKB1 P19838 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11517611 0.89 AKR1B1 (0.53) AKR1B1PTGS2KMT2ASMN1; SMN2DRD1
SCHEMBL11519465 0.89 AKR1B1 (0.69) AKR1B1PTGS2OPRK1PDE4DAKR1C3
SCHEMBL11520301 0.88 AKR1B1 (0.68) AKR1B1PTGS2OPRK1PDE4DAKR1C3
SCHEMBL11517083 0.86 AKR1B1 (0.72) AKR1B1PTGS2OPRK1PDE4DAKR1C3
SCHEMBL11519016 0.84 AKR1B1 (0.46) AKR1B1KMT2ASMN1; SMN2DRD1MEN1
SCHEMBL11519560 0.81 AKR1B1 (0.45) AKR1B1KMT2ADRD1MEN1PKM
SCHEMBL11520715 0.80 AKR1B1 (1.00) AKR1B1PTGS2OPRK1PDE4DAKR1C3
SCHEMBL11521696 0.79 AKR1B1 (0.76) AKR1B1PTGS2OPRK1PDE4DAKR1C3
SCHEMBL11518158 0.79 PGR (0.47) AKR1B1PDE4DKMT2ATP53SMN1; SMN2
SCHEMBL11517481 0.78 AKR1B1 (0.55) AKR1B1PTGS2PDE4DKMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172949-A 2,4-Disubstituted-5-oxo-5H-dibenzo[a,d]cycloheptenes SYNTEX (U.S.A.) INC. (US) 1979-10-30 US disclosed