SCHEMBL11520128

SCHEMBL11520128

NCc1c(CC(=O)O)cc(F)c(F)c1F

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 1/20 0.38
CXCL8 P10145 2/20 0.36
TSHR P16473 1/20 0.34
AKR1B1 P15121 2/20 0.33
CFD P00746 2/20 0.33
PTGS2 P35354 1/20 0.33
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
PTGS1 P23219 1/20 0.32
MCL1 Q07820 1/20 0.32
PLAU P00749 2/20 0.32
PLG P00747 1/20 0.31
F11 P03951 1/20 0.31
KLKB1 P03952 1/20 0.31
F7 P08709 1/20 0.31
TPSB2 P20231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30428405 0.79 CXCL8 (0.41) CXCL8TSHRAKR1B1CES2CES1
SCHEMBL7249684 0.79 CXCL8 (0.41) CXCL8TSHRAKR1B1CES2CES1
SCHEMBL15092154 0.76 AKR1B1 (0.41) CXCL8TSHRAKR1B1CES2CES1
SCHEMBL29009868 0.75 CA1 (0.40) AKR1B1CES2CES1
SCHEMBL3416130 0.74 PTGS1 (0.44) CXCL8TSHRPTGS2PTGS1
SCHEMBL3416138 0.70 AGBL2 (0.42)
SCHEMBL5062588 0.70 PTGS1 (0.40) CXCL8TSHRPTGS2PTGS1
SCHEMBL332576 0.70 CXCL8 (0.43) CXCL8TSHRAKR1B1
SCHEMBL29362137 0.70 CXCL8 (0.43) CXCL8TSHRAKR1B1
SCHEMBL11269548 0.70 CA1 (0.43) AKR1B1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed