SCHEMBL11524972

SCHEMBL11524972

CCOC(=O)C1=C(C)NC(CN)=C(C(=O)OCC)C1c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.71
KDM4E B2RXH2 6/20 0.60
ALDH1A1 P00352 4/20 0.60
TSHR P16473 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
ABCC1 P33527 1/20 0.59
GAA P10253 2/20 0.58
HSD17B10 Q99714 2/20 0.58
HPGD P15428 2/20 0.58
LMNA P02545 1/20 0.58
CASP1 P29466 1/20 0.55
CACNA1D Q01668 3/20 0.55
CACNA1F O60840 2/20 0.55
CACNA1S Q13698 2/20 0.55
CACNA1C Q13936 2/20 0.55
DHFR P00374 1/20 0.54
CACNA1B Q00975 1/20 0.53
MEN1 O00255 1/20 0.52
MAPT P10636 1/20 0.52
XBP1 P17861 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3027412 0.89 ADORA3 (0.89) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11729428 0.87 ADORA3 (0.68) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11521734 0.87 KDM4E (0.61) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11524242 0.87 KDM4E (0.59) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11524111 0.86 KDM4E (0.81) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11452070 0.86 ADORA3 (0.67) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL11522715 0.85 ABCC1 (0.58) ADORA3TSHRABCC1LMNACACNA1D
SCHEMBL11521974 0.85 TSHR (0.62) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL7286944 0.85 ADORA3 (0.65) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2
SCHEMBL29173863 0.85 ADORA3 (0.82) ADORA3KDM4EALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4177278-A 2-Alkyleneaminodihydropyridines compounds, their production and their medicinal use BAYER AKTIENGESELLSCHAFT (DE) 1979-12-04 US disclosed