SCHEMBL11526151

SCHEMBL11526151

N#Cc1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c2nc(Cl)nc(N)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 3/20 0.56
DOT1L Q8TEK3 3/20 0.56
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
PAX8 Q06710 2/20 0.51
HIF1A Q16665 1/20 0.51
ADORA3 P0DMS8 5/20 0.48
ADORA2A P29274 2/20 0.48
ADORA1 P30542 2/20 0.48
PDE2A O00408 1/20 0.48
ADRA1A P35348 1/20 0.48
PDE4D Q08499 1/20 0.48
PDE3A Q14432 1/20 0.48
PRMT5 O14744 1/20 0.47
PRMT3 O60678 1/20 0.47
DNMT1 P26358 1/20 0.47
EHMT2 Q96KQ7 1/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.46
GALR3 O60755 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18486808 0.87 DOT1L (0.56) ADKDOT1LLMNATP53PAX8
SCHEMBL18483493 0.87 DOT1L (0.56) ADKDOT1LLMNATP53PAX8
SCHEMBL18483516 0.85 DOT1L (0.54) ADKDOT1LPAX8HIF1APRMT5
SCHEMBL1738396 0.85 ADK (0.51) ADKDOT1LLMNATP53PAX8
SCHEMBL6727268 0.85 ADK (0.51) ADKDOT1LLMNATP53PAX8
SCHEMBL6737734 0.85 ADK (0.51) ADKDOT1LLMNATP53PAX8
SCHEMBL1738360 0.85 ADK (0.51) ADKDOT1LLMNATP53PAX8
SCHEMBL11529405 0.85 HIF1A (0.51) ADKDOT1LLMNATP53PAX8
SCHEMBL19101800 0.83 ADK (0.52) ADKDOT1LPAX8HIF1AADORA2A
SCHEMBL18483513 0.83 ADK (0.52) ADKDOT1LPAX8HIF1AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4140851-A Synthesis and antitumor activity of 2,4,5-trisubstituted-pyrrolo2,3-d]-pyrimidine nucleosides THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1979-02-20 US claimed
US-4140851-A Synthesis and antitumor activity of 2,4,5-trisubstituted-pyrrolo2,3-d]-pyrimidine nucleosides THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1979-02-20 US disclosed