SCHEMBL11527558

SCHEMBL11527558

CCOC(=O)N1CCN(C2=Nc3cc(F)ccc3Nc3ccsc32)CC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.49
HRH1 P35367 1/20 0.49
PAK1 Q13153 1/20 0.49
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
MAPT P10636 3/20 0.45
MAPK1 P28482 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11533130 0.86 MEN1 (0.52) CHRM1HRH1NOS3NOS1NOS2
SCHEMBL11531571 0.83 CHRM1 (0.52) CHRM1HRH1PAK1MAPTMAPK1
SCHEMBL11533744 0.80 CHRM1 (0.55) CHRM1HRH1PAK1
SCHEMBL11526082 0.79 CHRM1 (0.53) CHRM1HRH1PAK1
SCHEMBL11530525 0.77 DRD2 (0.51) CHRM1HRH1PAK1
SCHEMBL5477914 0.71 DRD2 (0.67) CHRM1HRH1MAPTMAPK1LMNA
SCHEMBL11532012 0.70 CHRM1 (0.66) CHRM1HRH1PAK1MAPTMAPK1
SCHEMBL11530539 0.69 CHRM1 (0.62) CHRM1HRH1PAK1
SCHEMBL11536340 0.69 CHRM1 (0.56) CHRM1HRH1PAK1MAPTKDM4E
SCHEMBL2036762 0.69 DRD2 (0.67) CHRM1HRH1MAPTMAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4172831-A CENTRAL NERVOUS SYSTEM LILLY INDUSTRIES LIMITED (GB) 1979-10-30 US disclosed
US-4115568-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed
US-4115574-A CNS ACTIVITY LILLY INDUSTRIES LIMITED (GB) 1978-09-19 US disclosed