SCHEMBL11528229

SCHEMBL11528229

OCc1cc2n(n1)-c1ccc(Cl)cc1C(c1ccccc1)=NC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 7/20 0.53
GABRA1 P14867 2/20 0.53
GABRA5 P31644 2/20 0.53
GABRA3 P34903 2/20 0.53
GABRA2 P47869 2/20 0.53
GABRB2 P47870 2/20 0.53
GABRP O00591 1/20 0.53
GABRD O14764 1/20 0.53
CACNA1F O60840 1/20 0.53
ALB P02768 1/20 0.53
GABRB1 P18505 1/20 0.53
GABRG2 P18507 1/20 0.53
GABRB3 P28472 1/20 0.53
AKR1C3 P42330 1/20 0.53
GABRA4 P48169 1/20 0.53
AKR1C2 P52895 1/20 0.53
GABRE P78334 1/20 0.53
CACNA1D Q01668 1/20 0.53
AKR1C1 Q04828 1/20 0.53
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11525923 0.83 OPRK1 (0.58) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11525787 0.83 OPRK1 (0.55) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL29833338 0.83 OPRK1 (0.55) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11526604 0.82 LMNA (0.59) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11525200 0.81 OPRK1 (0.53) OPRK1GABRA1GABRA5GABRA3GABRA2
Hydrochloric Acid SCHEMBL11527447 0.81 OPRK1 (0.53) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11523981 0.81 OPRK1 (0.55) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11446782 0.80 OPRK1 (0.55) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11526461 0.79 OPRK1 (0.54) OPRK1GABRA1GABRA5GABRA3GABRA2
SCHEMBL11526770 0.78 OPRK1 (0.53) OPRK1GABRA1GABRA5GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4157331-A SEDATIVES, TRANQUILIZERS, ANTICONVULSANTS, MUSCLE RELAXANTS HOFFMANN-LA ROCHE INC. (US) 1979-06-05 US disclosed
US-4153799-A ANXIOLYTICS, SEDATIVES, ANTICONVULSANTS, MUSCLE RELAXANTS, PYRAZOLE INTERMEDIATES HOFFMANN-LA ROCHE INC. (US) 1979-05-08 US disclosed
US-4130716-A ANXIOLYTICS, SEDATIVE, MUSCLE RELAXANT, ANTICONVULSANT HOFFMANN-LA ROCHE INC. (US) 1978-12-19 US disclosed