SCHEMBL11528604

SCHEMBL11528604

CCOC(=O)c1nn[nH]c1S.[NaH].[NaH]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.42
KDM4E B2RXH2 4/20 0.42
TSHR P16473 1/20 0.42
POLB P06746 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP1A2 P05177 3/20 0.38
ALDH1A1 P00352 2/20 0.38
ILK Q13418 1/20 0.38
TP53 P04637 1/20 0.37
ALOX12 P18054 1/20 0.37
DPP4 P27487 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
LMNA P02545 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23025720 0.80 PDE4D (0.50) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL7277080 0.79 PDE4D (0.44) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL1928112 0.79 PDE4D (0.44) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL5648877 0.79 KDM4E (0.46) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL11368014 0.77 ALDH1A1 (0.50) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL5906562 0.77 PDE4D (0.43) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL15897055 0.77 PDE4D (0.43) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL5648880 0.76 KDM4E (0.47) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL1412491 0.76 PDE4D (0.42) PDE4DKDM4ETSHRPOLBMEN1
SCHEMBL1930598 0.75 PDE4D (0.41) PDE4DKDM4ETSHRPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4142046-A BACTERICIDES, 7-AMINO-CEPHALOSPORINS SMITHKLINE CORPORATION (US) 1979-02-27 US disclosed
US-4060610-A Pharmaceutical compositions comprising 7-acyl-3-(substituted triazolyl thiomethyl)-cephalosporins and methods of treating bacterial infections SMITHKLINE CORPORATION (US) 1977-11-29 US disclosed
US-3989694-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-11-02 US disclosed