SCHEMBL11529414

SCHEMBL11529414

CCOC(=O)C(C)C(=O)c1cnccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
KMT2A Q03164 1/20 0.48
POLB P06746 3/20 0.45
TSHR P16473 2/20 0.45
TP53 P04637 1/20 0.45
KDM4E B2RXH2 5/20 0.44
NAPRT Q6XQN6 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
HPGD P15428 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
MC4R P32245 1/20 0.43
ADRA1A P35348 1/20 0.43
MC3R P41968 1/20 0.43
RECQL P46063 1/20 0.43
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11529446 0.86 NPC1 (0.49) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL5578127 0.84 KDM4E (0.47) SMN1; SMN2NPC1RAB9AKMT2ATSHR
SCHEMBL11527512 0.83 RAB9A (0.50) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL3400596 0.83 NPC1 (0.47) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11529880 0.83 NPC1 (0.47) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11529442 0.82 NPC1 (0.46) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11529156 0.81 RAB9A (0.45) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11529222 0.80 NPC1 (0.44) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11530272 0.79 POLB (0.49) SMN1; SMN2NPC1RAB9AKMT2APOLB
SCHEMBL11526544 0.79 KDM4E (0.46) SMN1; SMN2NPC1RAB9AKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7288652-B2 Reacting methyl 2-methyl-3-(pyrazin-2-yl)-3-oxopropionate with phosphorus pentasulfide in presence of mixed solvent of toluene andxylene under reflux to produce an oltipraz crude crystal; recrystallization; sulfiding, cyclization CJ CORPORATION (KR) 2007-10-30 US disclosed
US-7288652-B2 Reacting methyl 2-methyl-3-(pyrazin-2-yl)-3-oxopropionate with phosphorus pentasulfide in presence of mixed solvent of toluene andxylene under reflux to produce an oltipraz crude crystal; recrystallization; sulfiding, cyclization CJ CORPORATION (KR) 2007-10-30 US disclosed
US-4144339-A TREATMENT OF BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1979-03-13 US disclosed
US-4138487-A NEMATOCIDES RHONE-POULENC INDUSTRIES (FR) 1979-02-06 US disclosed
US-4110450-A BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1978-08-29 US disclosed