SCHEMBL11533784

SCHEMBL11533784

Cc1cnc(S(C)(=O)=O)o1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.40
PIK3CG P48736 1/20 0.40
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28980204 0.76 PIK3CA (0.36) PIK3CAPIK3CG
SCHEMBL21899214 0.74 PIK3CA (0.35) PIK3CAPIK3CG
SCHEMBL27892601 0.72 NOTUM (0.37) PIK3CAPIK3CG
SCHEMBL11528398 0.72 PIK3CA (0.35) PIK3CAPIK3CG
SCHEMBL9700791 0.71 LOXL2 (0.34) PIK3CAPIK3CG
SCHEMBL3464438 0.67 PIK3CA (0.37) PIK3CAPIK3CG
SCHEMBL31304016 0.66 NOTUM (0.49) PIK3CAPIK3CGCA12CA1CA2
SCHEMBL30580704 0.66 PTGS2 (0.43) PIK3CAPIK3CGCA12CA1CA2
SCHEMBL17796279 0.65
SCHEMBL27876055 0.65 KLKB1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198710-A1 PHARMACEUTICAL COMPOSITIONS AND COMBINATIONS COMPRISING INHIBITORS OF THE ANDROGEN RECEPTOR AND USES THEREOF ESSA PHARMA, INC. (CA) 2020-10-01 WO disclosed
US-4143047-A 2-SULFINYL AND 2-SULFONYL OXAZOLES LILLY INDUSTRIES LIMITED (GB) 1979-03-06 US disclosed