SCHEMBL11534820

SCHEMBL11534820

Cc1[c]c(C(N)=O)cc(C)c1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.36
TPMT P51580 1/20 0.33
PRSS1 P07477 1/20 0.32
PRSS2 P07478 1/20 0.32
C1S P09871 1/20 0.32
PRSS3 P35030 1/20 0.32
PARP10 Q53GL7 1/20 0.32
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
NNMT P40261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1637046 0.80 TPMT (0.34) TPMT
SCHEMBL28912366 0.80 TPMT (0.44) TPMTKDM4E
SCHEMBL1636895 0.71
SCHEMBL1971878 0.70 PARP1 (0.45) PARP1PARP10CYP3A4
SCHEMBL18896 0.69
SCHEMBL4926679 0.68 SIRT3 (0.37) NNMT
SCHEMBL28817336 0.67 CYP3A4 (0.41) PARP1PRSS1PRSS2PRSS3PARP10
SCHEMBL23531515 0.67 ALDH1A1 (0.37)
SCHEMBL9982849 0.67 ALDH1A1 (0.37)
SCHEMBL3888279 0.67 ALDH1A1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4137325-A Antisecretory oxamic acid esters AMERICAN HOME PRODUCTS CORPORATION (US) 1979-01-30 US claimed
CN-108137532-A PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV保健英国第五有限公司 2018-06-08 CN disclosed
US-4137325-A Antisecretory oxamic acid esters AMERICAN HOME PRODUCTS CORPORATION (US) 1979-01-30 US disclosed