SCHEMBL11535490

SCHEMBL11535490

CC(C)N(CCC(C#N)(CCN1CCCCCC1)c1ccccc1F)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 2/20 0.43
CYP2D6 P10635 3/20 0.35
MAPK1 P28482 1/20 0.35
PKM P14618 1/20 0.35
LMNA P02545 1/20 0.34
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
CHRM1 P11229 1/20 0.34
OPRM1 P35372 1/20 0.34
KCNH2 Q12809 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11532343 1.00 KCNA3 (0.43) KCNA3CYP2D6MAPK1PKMLMNA
SCHEMBL11530765 0.99 KCNA3 (0.41) KCNA3CYP2D6MAPK1PKMLMNA
SCHEMBL11533327 0.87 KCNA3 (0.43) KCNA3CYP2D6MAPK1LMNACHRM2
SCHEMBL11531523 0.86 CYP3A4 (0.34) CYP2D6CHRM2CHRM1OPRM1KCNH2
SCHEMBL11486857 0.85 KCNA3 (0.41) KCNA3CYP2D6MAPK1LMNAALDH1A1
SCHEMBL11534012 0.84 KCNA3 (0.55) KCNA3CYP2D6MAPK1LMNACHRM2
SCHEMBL11533521 0.84 KCNA3 (0.55) KCNA3CYP2D6MAPK1LMNACHRM2
SCHEMBL11486790 0.84 HRH3 (0.37) LMNACHRM2ALDH1A1RAB9ANPSR1
SCHEMBL11539299 0.83 KCNA3 (0.53) KCNA3CYP2D6MAPK1LMNACHRM2
SCHEMBL11537461 0.82 KCNA3 (0.41) KCNA3CYP2D6MAPK1ALDH1A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4153797-A α-Aryl-α, α-bis[ω- (disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1979-05-08 US disclosed
US-4107205-A α-Aryl-α,α-bis[ω-(disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1978-08-15 US disclosed