SCHEMBL11536976

SCHEMBL11536976

Cc1nnc2sc3ccccc3n12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.66
PDGFRA P16234 1/20 0.66
CDK5 Q00535 1/20 0.66
DYRK1A Q13627 1/20 0.66
LRRK2 Q5S007 1/20 0.66
CLK4 Q9HAZ1 1/20 0.66
DYRK1B Q9Y463 1/20 0.66
ALDH1A1 P00352 3/20 0.55
RECQL P46063 1/20 0.51
GAA P10253 1/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
KDM4E B2RXH2 2/20 0.49
PARP2 Q9UGN5 3/20 0.47
TNKS2 Q9H2K2 2/20 0.47
RAB9A P51151 4/20 0.47
NPC1 O15118 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
POLB P06746 2/20 0.47
TSHR P16473 2/20 0.47
HSD17B10 Q99714 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11747896 0.98 CHEK1 (0.64) CHEK1PDGFRACDK5DYRK1ALRRK2
Acetic Acid SCHEMBL11746162 0.92 CHEK1 (0.57) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11739724 0.82 ALDH1A1 (0.60) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11534080 0.79 PARP2 (0.55) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11536264 0.79 PARP10 (0.73) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11741753 0.78 CHEK1 (0.66) CHEK1PDGFRACDK5DYRK1ALRRK2
Bromide SCHEMBL11743370 0.78 CHEK1 (0.96) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11746931 0.78 CHEK1 (0.66) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11744129 0.78 CHEK1 (0.66) CHEK1PDGFRACDK5DYRK1ALRRK2
SCHEMBL11743929 0.78 CHEK1 (0.66) CHEK1PDGFRACDK5DYRK1ALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4064261-A TRIAZOLOBENOXAZOLE, TRIAZOLOBENZOTHIAZOLE COMPOUNDS ELI LILLY AND COMPANY (US) 1977-12-20 US claimed
US-3937713-A Process for the preparation of s-triazolo[3,4-b]benzothiazoles ELI LILLY AND COMPANY (US) 1976-02-10 US claimed
US-4134914-A 1-Acyl-4-substituted phenyl thiosemicarbazides ELI LILLY AND COMPANY (US) 1979-01-16 US disclosed
US-4082762-A 4-(2-HALOPHENYL)-1,2,4-TRIAZOLE-3-THIOL COMPOUNDS ELI LILLY AND COMPANY (US) 1978-04-04 US disclosed
US-4064261-A TRIAZOLOBENOXAZOLE, TRIAZOLOBENZOTHIAZOLE COMPOUNDS ELI LILLY AND COMPANY (US) 1977-12-20 US disclosed
US-3937713-A Process for the preparation of s-triazolo[3,4-b]benzothiazoles ELI LILLY AND COMPANY (US) 1976-02-10 US disclosed