SCHEMBL11537656

SCHEMBL11537656

CCCOc1cccc(C(c2ccccc2)(c2ccccc2)c2ccc(C#N)nc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
LMNA P02545 2/20 0.36
FGFR1 P11362 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.36
CYSLTR1 Q9Y271 1/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
ACACB O00763 1/20 0.36
KAT6A Q92794 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11539449 0.82 KMT2A (0.41) KMT2AMAPTSMN1; SMN2L3MBTL1LMNA
SCHEMBL11536344 0.82 KIF11 (0.38) KMT2AMEN1
SCHEMBL11533562 0.79 CHEK1 (0.43) MAPTALDH1A1TSHR
SCHEMBL11536087 0.79 KMT2A (0.50) KMT2AMAPTSMN1; SMN2L3MBTL1LMNA
SCHEMBL11539601 0.79 NPC1 (0.40) KMT2AMAPTPOLBNPC1ALDH1A1
SCHEMBL11538842 0.78 KMT2A (0.45) KMT2AMAPTSMN1; SMN2LMNAHTT
SCHEMBL11536609 0.76 CHEK1 (0.38) KMT2AMEN1
SCHEMBL11536728 0.76 CHEK1 (0.35) SMN1; SMN2NPC1RAB9ATSHR
SCHEMBL11536969 0.76 CHEK1 (0.38) SMN1; SMN2ALDH1A1TSHR
SCHEMBL11534250 0.74 CHEK1 (0.49) MAPTL3MBTL1CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed