SCHEMBL11539849

SCHEMBL11539849

CC(C)(C)C(=O)OC(COc1cccc2[nH]ncc12)CN1CCC(COc2ccccc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 7/20 0.41
DRD2 P14416 2/20 0.39
P2RY1 P47900 2/20 0.38
ADRB2 P07550 5/20 0.37
ADRB1 P08588 5/20 0.37
ADRB3 P13945 5/20 0.37
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
ABCB1 P08183 2/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11539450 0.87 ADRB2 (0.47) DRD4ADRB2ADRB1ADRB3
SCHEMBL11539298 0.86 P2RY1 (0.39) DRD4DRD2P2RY1ADRB2ADRB1
Hydrochloric Acid SCHEMBL11544679 0.85 P2RY1 (0.39) DRD4DRD2P2RY1ADRB2ADRB1
SCHEMBL11541245 0.85 HTR3A (0.40) DRD4P2RY1ADRB2ADRB1ADRB3
Hydrochloric Acid SCHEMBL11541081 0.84 HTR3A (0.39) DRD4P2RY1ADRB2ADRB1ADRB3
SCHEMBL11537535 0.83 DRD4 (0.56) DRD4DRD2ADRB2ADRB1ADRB3
Hydrochloric Acid SCHEMBL11372638 0.82 ADRB2 (0.43) DRD4P2RY1ADRB2ADRB1ADRB3
SCHEMBL11541253 0.82 DRD4 (0.38) DRD4P2RY1CARM1PRMT6ABCB1
Hydrochloric Acid SCHEMBL11541088 0.81 P2RY1 (0.38) DRD4P2RY1CARM1PRMT6ABCB1
SCHEMBL6295417 0.78 ADRB2 (0.49) DRD4ADRB2ADRB1ADRB3ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4146630-A HYPOTENSIVE AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1979-03-27 US disclosed