SCHEMBL11540482

SCHEMBL11540482

CCOC1(c2ccccc2)CCN(C(=O)CC2COc3ccccc3O2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 1/20 0.45
GLA P06280 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
OPRL1 P41146 1/20 0.44
HTT P42858 1/20 0.44
HPGD P15428 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11537590 0.87 KDM4E (0.45) DRD2KDM4EGAAMEN1KMT2A
SCHEMBL11537204 0.84 LTA4H (0.52) DRD2KDM4EGAAPOLBHTT
Maleic Acid SCHEMBL11534674 0.81 DRD2 (0.45) DRD2KDM4EGAAMEN1MAPT
Fumaric Acid SCHEMBL11534679 0.81 DRD2 (0.45) DRD2KDM4EGAAMEN1MAPT
SCHEMBL3257424 0.73 MEN1 (0.62) KDM4EGAAMEN1GLAMAPT
SCHEMBL11538594 0.73 HTT (0.58) DRD2KDM4EGAAMAPTPOLB
Hydrochloric Acid SCHEMBL11537492 0.72 DRD3 (0.55) DRD2KDM4EGAAMAPTOPRM1
SCHEMBL9692477 0.70 CYP1A2 (0.63) GAAMEN1GLAMAPTKMT2A
SCHEMBL4553361 0.70 HTT (0.71) MEN1KMT2APOLBHTTHPGD
SCHEMBL11535627 0.70 DRD2 (0.50) DRD2MEN1KMT2AOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4140781-A Analgesic and neuraleptic 2-piperidinoalkyl-1,4-benzodioxans CIBA-GEIGY CORPORATION (US) 1979-02-20 US disclosed
US-4129655-A Neuroleptic 2-piperidinoalkyl-1,4-benzodioxans CIBA-GEIGY CORPORATION (US) 1978-12-12 US disclosed
US-4104396-A NEUROLEPTIC, ANALGESIC CIBA-GEIGY CORPORATION (US) 1978-08-01 US disclosed