SCHEMBL11544247

SCHEMBL11544247

CC(C)(C)N1Cc2c(Cl)cccc2C(c2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 8/20 0.48
SLC6A4 P31645 8/20 0.48
SLC6A3 Q01959 8/20 0.48
LMNA P02545 2/20 0.47
MAPK1 P28482 2/20 0.47
RGS12 O14924 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
ALOX12 P18054 1/20 0.47
NFKB1 P19838 1/20 0.47
HTR2A P28223 1/20 0.47
ADRA1A P35348 1/20 0.47
PTGS2 P35354 1/20 0.47
HRH1 P35367 1/20 0.47
OPRM1 P35372 1/20 0.47
GNAI1 P63096 1/20 0.47
KCNH2 Q12809 1/20 0.47
KIF11 P52732 3/20 0.44
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027703 0.81 SLC6A2 (0.71) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL11921529 0.68 SLC6A2 (0.68) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL24352150 0.66 HRH3 (0.35) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL4030851 0.65 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL2568332 0.65 SLC9A3 (0.67) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL11101484 0.64 SLC6A2 (0.59) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL25452943 0.64 ADRA2A (0.57) LMNACYP1A2CYP2D6HTR2AADRA1A
SCHEMBL22024397 0.64 KIF11 (0.36) SLC6A2SLC6A4SLC6A3LMNAMAPK1
SCHEMBL16835251 0.64 HTR2C (0.61) MAPK1CYP1A2CYP3A4CYP2D6NFKB1
SCHEMBL4027936 0.64 SLC6A2 (0.71) SLC6A2SLC6A4SLC6A3LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4175191-A 4-Phenyl isoquinolines SANDOZ, INC. (US) 1979-11-20 US disclosed
US-3989704-A 3-Substituted-4-aryl isoquinolines SANDOZ, INC. (US) 1976-11-02 US disclosed