SCHEMBL11544834

SCHEMBL11544834

O=C(O)c1cc(N2CCCC2)c(Oc2ccccc2)c(S(=O)(=O)Cl)c1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.79
HSD17B10 Q99714 4/20 0.79
ALDH1A1 P00352 4/20 0.79
LMNA P02545 4/20 0.79
HPGD P15428 3/20 0.79
USP2 O75604 2/20 0.79
HIF1A Q16665 2/20 0.79
SLC6A4 P31645 1/20 0.79
ERAP1 Q9NZ08 4/20 0.43
ERAP2 Q6P179 1/20 0.43
TSHR P16473 2/20 0.41
POLB P06746 2/20 0.41
CA2 P00918 1/20 0.40
BLM P54132 1/20 0.40
SLC12A2 P55011 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
GAA P10253 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11542238 0.89 ALDH1A1 (0.63) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL49473 0.88 KDM4E (1.00) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL1741994 0.88 KDM4E (1.00) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL30230376 0.88 KDM4E (1.00) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL9837127 0.87 KDM4E (0.98) KDM4EHSD17B10ALDH1A1LMNAHPGD
SCHEMBL2741891 0.87 KDM4E (0.98) KDM4EHSD17B10ALDH1A1LMNAHPGD
SCHEMBL14879729 0.87 KDM4E (0.77) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL7895002 0.86 KDM4E (0.95) KDM4EHSD17B10ALDH1A1LMNAHPGD
Piretanide SCHEMBL18075706 0.86 KDM4E (0.95) KDM4EHSD17B10ALDH1A1LMNAHPGD
SCHEMBL11542770 0.86 KDM4E (0.95) KDM4EHSD17B10ALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4161531-A Diuretic and saluretic 5-sulfamoylbenzoic acid derivatives carrying a heterocyclic substituent HOECHST AKTIENGESELLSCHAFT (DE) 1979-07-17 US disclosed
US-4118397-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US disclosed
US-4111953-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DE) 1978-09-05 US disclosed
US-4093735-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DT) 1978-06-06 US disclosed
US-4010273-A DIURETICS, SALURETICS HOECHST AKTIENGESELLSCHAFT (DT) 1977-03-01 US disclosed