SCHEMBL11546340

SCHEMBL11546340

COC(=O)Nc1ccc(C(=O)CBr)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.45
HPGD P15428 2/20 0.45
PDK1 Q15118 3/20 0.44
PDK2 Q15119 3/20 0.44
PDK3 Q15120 3/20 0.44
PDK4 Q16654 3/20 0.44
PTPN1 P18031 1/20 0.41
EGFR P00533 2/20 0.40
KDR P35968 2/20 0.40
MAPT P10636 2/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16753317 0.82 HDAC1 (0.46) GSK3BHPGDPTPN1MAPTALDH1A1
SCHEMBL11547679 0.81 HPGD (0.50) HPGDPDK1PDK2PDK3PDK4
SCHEMBL11552737 0.81 GSK3B (0.42) GSK3BHPGDPTPN1MAPTUSP2
SCHEMBL2089909 0.76 HPGD (0.70) HPGDMAPTTAS1R3TAS1R1TAS1R2
SCHEMBL2095473 0.76 HPGD (0.58) HPGDPDK1PDK2PDK3PDK4
SCHEMBL31386348 0.76 GSK3B (0.47) GSK3BHPGDPDK2PDK4PTPN1
SCHEMBL11547384 0.75 GSK3B (0.37) GSK3BHPGDMAPTUSP2ALDH1A1
SCHEMBL29620782 0.75 GSK3B (0.54) GSK3BMAPTTAS1R3TAS1R1ALDH1A1
SCHEMBL2166529 0.75 GSK3B (0.54) GSK3BMAPTTAS1R3TAS1R1ALDH1A1
SCHEMBL19170620 0.74 MAPT (0.57) HPGDEGFRKDRMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4145363-A ANTIASTHMATICS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1979-03-20 US disclosed
US-4063025-A PROPHYLAXIS, ANTIASTHMATIC YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1977-12-13 US disclosed