SCHEMBL8596134

SCHEMBL8596134

COc1ccc2c(C(=O)c3ccc(OCCN(C)C)cc3)c(-c3ccccc3)sc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.60
ESR2 Q92731 13/20 0.60
CNR1 P21554 1/20 0.57
CNR2 P34972 1/20 0.57
ITGA4 P13612 1/20 0.55
NAPEPLD Q6IQ20 1/20 0.55
PAX8 Q06710 1/20 0.54
HCRTR1 O43613 1/20 0.53
TUBB4A P04350 1/20 0.53
TUBB P07437 1/20 0.53
TUBA3C P0DPH7 1/20 0.53
TUBA1B P68363 1/20 0.53
TUBA4A P68366 1/20 0.53
TUBB4B P68371 1/20 0.53
TUBB3 Q13509 1/20 0.53
TUBB2A Q13885 1/20 0.53
TUBB8 Q3ZCM7 1/20 0.53
TUBA3E Q6PEY2 1/20 0.53
TUBA1A Q71U36 1/20 0.53
TUBA1C Q9BQE3 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11548759 0.95 ESR1 (0.66) ESR1ESR2CNR1CNR2ITGA4
SCHEMBL11555855 0.94 ESR1 (0.68) ESR1ESR2CNR1CNR2ITGA4
SCHEMBL8597235 0.90 ESR1 (0.58) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL11552316 0.90 ESR1 (0.61) ESR1ESR2CNR1CNR2PAX8
SCHEMBL7626639 0.90 ESR1 (0.67) ESR1ESR2CNR1
SCHEMBL4652009 0.89 CNR2 (0.75) ESR1ESR2CNR1CNR2ITGA4
SCHEMBL8600465 0.88 ESR1 (0.62) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL8599094 0.87 ESR1 (0.58) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL11547336 0.87 ESR1 (0.61) ESR1ESR2CNR1CNR2TUBB4A
SCHEMBL11550720 0.86 CNR1 (0.67) ESR1ESR2CNR1CNR2ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641791-B1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG CO LTD (JP) 1998-01-28 EP disclosed
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
EP-0641791-A1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-03-08 EP disclosed