SCHEMBL11552115

SCHEMBL11552115

C=CCN1C(=O)CC(=O)N(c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.62
PDE4D Q08499 1/20 0.62
PTGDR2 Q9Y5Y4 4/20 0.45
HPGD P15428 1/20 0.40
CCKBR P32239 1/20 0.38
CASP6 P55212 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 2/20 0.36
ALDH2 P05091 2/20 0.36
HTT P42858 1/20 0.36
KMO O15229 1/20 0.36
ALOX12 P18054 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRM1 P11229 1/20 0.35
ALDH3A1 P30838 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11550187 0.84 OPRK1 (0.66) OPRK1PDE4DPTGDR2HPGDCASP6
SCHEMBL11552056 0.84 OPRK1 (0.70) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11776339 0.81 OPRK1 (0.67) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11754667 0.81 OPRK1 (0.70) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11554122 0.81 OPRK1 (0.62) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11776991 0.81 OPRK1 (0.65) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11550773 0.81 OPRK1 (0.62) OPRK1PDE4DHPGDCCKBRCASP6
SCHEMBL11434574 0.80 OPRK1 (0.51) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11761654 0.80 OPRK1 (0.67) OPRK1PDE4DPTGDR2HPGDCCKBR
SCHEMBL11778247 0.80 OPRK1 (0.64) OPRK1PDE4DPTGDR2HPGDCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4001408-A SUBSTITUTED HETEROCYCLIC COMPOUNDS, PROCESSES AND COMPOSITION INCLUDING THOSE ROUSSEL-UCLAF (FR) 1977-01-04 US claimed
US-3984398-A 1,5-Benzodiazepine-2,4-diones ROUSSEL-UCLAF (FR) 1976-10-05 US claimed
US-4138572-A Malonanilic derivatives ROUSSEL UCLAF (FR) 1979-02-06 US disclosed
US-4001408-A SUBSTITUTED HETEROCYCLIC COMPOUNDS, PROCESSES AND COMPOSITION INCLUDING THOSE ROUSSEL-UCLAF (FR) 1977-01-04 US disclosed
US-3984398-A 1,5-Benzodiazepine-2,4-diones ROUSSEL-UCLAF (FR) 1976-10-05 US disclosed